SCHEMBL7260689

SCHEMBL7260689

CCOC(=O)C(Cc1ccc(O)cc1)NC(=O)OC(C)(C)C

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSS P25774 6/20 0.63
CTSK P43235 5/20 0.63
CYP1A2 P05177 1/20 0.51
CYP2C9 P11712 1/20 0.51
CYP2C19 P33261 1/20 0.51
HTT P42858 1/20 0.51
LY96 Q9Y6Y9 1/20 0.51
ALDH1A1 P00352 3/20 0.50
MAPT P10636 3/20 0.50
CTSL P07711 1/20 0.50
CTSB P07858 1/20 0.50
ITGB3 P05106 1/20 0.48
ITGA2B P08514 1/20 0.48
ACE P12821 1/20 0.48
KLK5 Q9Y337 1/20 0.47
TACR1 P25103 1/20 0.47
KDM4E B2RXH2 1/20 0.47
GAA P10253 1/20 0.47
PKM P14618 1/20 0.47
HPGD P15428 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL920111 1.00 CTSS (0.63) CTSSCTSKCYP1A2CYP2C9CYP2C19
SCHEMBL20045974 0.91 PPARG (0.53) CTSSCTSKCYP1A2CYP2C9CYP2C19
SCHEMBL14803767 0.91 PPARG (0.53) CTSSCTSKCYP1A2CYP2C9CYP2C19
SCHEMBL14405376 0.91 CTSS (0.67) CTSSCTSKLY96MAPTCTSL
SCHEMBL2076110 0.91 CTSS (0.67) CTSSCTSKLY96MAPTCTSL
SCHEMBL309644 0.91 CTSS (0.67) CTSSCTSKLY96MAPTCTSL
SCHEMBL30374091 0.89 CTSS (0.66) CTSSCTSKLY96CTSLCTSB
SCHEMBL539574 0.89 CTSS (0.66) CTSSCTSKLY96CTSLCTSB
SCHEMBL2574440 0.89 CTSS (0.66) CTSSCTSKLY96CTSLCTSB
SCHEMBL539575 0.89 CTSS (0.66) CTSSCTSKLY96CTSLCTSB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 18 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260077069-A1 COMBINATIONS OF CONTRAST AGENTS BAYER AG (DE) 2026-03-19 US disclosed
EP-4583925-A1 COMBINATIONS OF CONTRAST AGENTS Bayer Aktiengesellschaft (DE) 2025-07-16 EP disclosed
EP-4584251-A1 NEW CONTRAST AGENTS FOR USE IN DIAGNOSTIC IMAGING Bayer Aktiengesellschaft (DE) 2025-07-16 EP disclosed
WO-2024052549-A1 NEW CONTRAST AGENTS FOR USE IN DIAGNOSTIC IMAGING BAYER AKTIENGESELLSCHAFT (DE) 2024-03-14 WO disclosed
WO-2024052573-A1 COMBINATIONS OF CONTRAST AGENTS BAYER AKTIENGESELLSCHAFT (DE) 2024-03-14 WO disclosed
EP-4335461-A1 COMBINATIONS OF CONTRAST AGENTS Bayer AG (DE) 2024-03-13 EP disclosed
EP-4335840-A1 NEW CONTRAST AGENTS FOR USE IN DIAGNOSTIC IMAGING Bayer Aktiengesellschaft (DE) 2024-03-13 EP disclosed
CN-111315746-B Tryptophan hydroxylase inhibitors and pharmaceutical compositions comprising the same 光州科学技术院 2022-11-29 CN disclosed
CN-114616229-A Tricyclic compounds and pharmaceutical uses thereof 镇斗生物科技股份公司 2022-06-10 CN disclosed
CN-113840825-A Aldose reductase inhibitors 应用治疗公司 2021-12-24 CN disclosed
CN-111315746-A Novel tryptophan hydroxylase inhibitors and pharmaceutical compositions comprising the same 光州科学技术院 2020-06-19 CN disclosed
CN-101948552-A Linear polystyrene-supported chiral oxazolidine-2-selenium ketone and preparation method thereof UNIV HUBEI 2011-01-19 CN disclosed
CN-101914174-A Linear polystyrene-supported (4S)-oxazolidine-2-benzimine as well as preparation method and application thereof UNIV HUBEI 2010-12-15 CN disclosed
CN-1301964-C Inhibitors of alpha 4-mediated cell adhesion TANABE SEIYAKU CO (JP) 2007-02-28 CN disclosed
US-6593338-B2 Inhibit the binding of integrins to their ligands and are of use in the prophylaxis and treatment of immuno or inflammatory disorders or disorders involving the inappropriate growth or migration of cells. CELLTECH R&D LIMITED (GB) 2003-07-15 US disclosed
US-20020137935-A1 3-Substituted 2,7-naphthyridin-1-yl derivatives CELLTECH R&D LIMITED (GB) 2002-09-26 US disclosed
CN-1288457-A Inhibitors of & alpha, 4 mediated cell adhesion TANABE SEIYAKU CO (JP) 2001-03-21 CN disclosed
CN-1098409-A 2-piperazinone compounds and application thereof TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1995-02-08 CN disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20020137935-A1 3-Substituted 2,7-naphthyridin-1-yl derivatives ITGB2, ICAM1, ITGB1 CTSS 2273/4885CTSK 3047/4885CYP1A2 999/4885
US-20260077069-A1 COMBINATIONS OF CONTRAST AGENTS GBA1, GBA3, GLS2 CTSS 386/4885CTSK 1543/4885CYP1A2 1646/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.