SCHEMBL7260927

SCHEMBL7260927

COCCc1cc2ccccc2c(=O)[nH]1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LOXL2 Q9Y4K0 1/20 0.58
KDM4E B2RXH2 4/20 0.53
GAA P10253 2/20 0.53
CDC25B P30305 10/20 0.46
THRB P10828 3/20 0.46
APAF1 O14727 6/20 0.44
CASP3 P42574 6/20 0.44
SENP8 Q96LD8 6/20 0.44
SENP7 Q9BQF6 6/20 0.44
SENP6 Q9GZR1 4/20 0.44
CASP6 P55212 4/20 0.44
TNKS O95271 2/20 0.44
ALDH1A1 P00352 4/20 0.43
SAE1 Q9UBE0 3/20 0.43
UBA2 Q9UBT2 3/20 0.43
HPGD P15428 3/20 0.43
MAPT P10636 2/20 0.43
UBE2I P63279 2/20 0.43
RECQL P46063 1/20 0.43
GALK1 P51570 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7343701 0.79 LOXL2 (0.60) LOXL2KDM4EGAACDC25BTHRB
SCHEMBL28566574 0.78 LOXL2 (0.55) LOXL2
SCHEMBL2599466 0.78 LOXL2 (0.74) LOXL2KDM4EGAACDC25BTHRB
SCHEMBL1720643 0.78 LOXL2 (0.68) LOXL2KDM4EGAACDC25BTHRB
SCHEMBL6646959 0.77 LOXL2 (0.58) LOXL2KDM4EGAACDC25BTHRB
SCHEMBL2532412 0.77 PARP1 (0.65) LOXL2KDM4EGAAAPAF1CASP3
SCHEMBL6603861 0.77 LOXL2 (0.62) LOXL2KDM4EGAACDC25BTHRB
SCHEMBL6647824 0.75 LOXL2 (0.55) LOXL2KDM4EGAACDC25BTHRB
SCHEMBL7946899 0.75 LOXL2 (0.55) LOXL2KDM4EGAACDC25BTHRB
SCHEMBL31386969 0.75 PARP1 (0.42) LOXL2KDM4ECDC25BTHRBTNKS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1284967-A1 3-SUBSTITUTED ISOQUINOLIN-1-YL DERIVATIVES Celltech R&D Limited (GB) 2003-02-26 EP disclosed
WO-2001092233-A1 3-SUBSTITUTED ISOQUINOLIN-1-YL DERIVATIVES CELLTECH R & D LIMITED (GB) 2001-12-06 WO disclosed