SCHEMBL7264349

SCHEMBL7264349

C=CC(=O)C(C/C=C/c1ccccc1)C(=O)O

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRIK1 P39086 4/20 0.51
GRIK2 Q13002 4/20 0.51
PAM P19021 1/20 0.49
HTR2A P28223 3/20 0.46
PIN1 Q13526 2/20 0.43
MAOB P27338 1/20 0.41
CYP1A2 P05177 2/20 0.41
CYP2C19 P33261 1/20 0.41
HDAC3 O15379 1/20 0.40
TNKS O95271 1/20 0.40
HDAC4 P56524 1/20 0.40
HDAC1 Q13547 1/20 0.40
HCAR2 Q8TDS4 1/20 0.40
HDAC7 Q8WUI4 1/20 0.40
HDAC2 Q92769 1/20 0.40
HDAC10 Q969S8 1/20 0.40
HDAC11 Q96DB2 1/20 0.40
HDAC8 Q9BY41 1/20 0.40
TNKS2 Q9H2K2 1/20 0.40
HDAC6 Q9UBN7 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7264360 1.00 GRIK1 (0.51) GRIK1GRIK2PAMHTR2APIN1
SCHEMBL27989732 0.88 GRIK1 (0.62) GRIK1GRIK2PAMHTR2APIN1
SCHEMBL27689553 0.88 GRIK1 (0.62) GRIK1GRIK2PAMHTR2APIN1
SCHEMBL6188960 0.79 GRIK1 (0.54) GRIK1GRIK2PAMHTR2APIN1
SCHEMBL6188957 0.79 GRIK1 (0.54) GRIK1GRIK2PAMHTR2APIN1
SCHEMBL13258634 0.77 GRIK1 (0.63) GRIK1GRIK2PAMHTR2ACYP2C19
SCHEMBL31506964 0.76 PAM (0.52) GRIK1GRIK2PAMHTR2APIN1
SCHEMBL5835825 0.75 GRIK1 (0.50) GRIK1GRIK2PAMHTR2APIN1
SCHEMBL5835829 0.75 GRIK1 (0.50) GRIK1GRIK2PAMHTR2APIN1
SCHEMBL4872078 0.75 GRIK1 (0.57) GRIK1GRIK2PAMHTR2APIN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6642035-B2 Synthesis of B-keto esters THE SCRIPPS RESEARCH INSTITUTE 2003-11-04 US disclosed
US-20020102671-A1 Synthesis of B-keto esters SCRIPPS RESEARCH INSTITUTE, THE 2002-08-01 US disclosed