SCHEMBL7266106

SCHEMBL7266106

CNC[C@H]1CC[C@H](c2nc3ccccc3[nH]2)CC1

nearest known ligand 0.60

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
GID4 Q8IVV7 2/20 0.51
IDO1 P14902 1/20 0.49
HTR2B P41595 2/20 0.48
POLB P06746 4/20 0.47
PKM P14618 2/20 0.46
MAPT P10636 2/20 0.45
HSD17B10 Q99714 1/20 0.45
NPY5R Q15761 1/20 0.44
ALDH1A1 P00352 1/20 0.44
HPGD P15428 1/20 0.44
TSHR P16473 1/20 0.44
KDM4E B2RXH2 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7266112 1.00 GID4 (0.51) GID4IDO1HTR2BPOLBPKM
SCHEMBL10177547 0.85 IDO1 (0.54) GID4IDO1HTR2BPOLBPKM
SCHEMBL2276872 0.83 ALDH1A1 (0.59) GID4IDO1HTR2BPOLBPKM
Hydrochloric Acid SCHEMBL31596380 0.82 MAPT (0.57) GID4HTR2BPOLBPKMMAPT
SCHEMBL5024041 0.81 IDO1 (0.52) GID4IDO1HTR2BPOLBPKM
SCHEMBL5024044 0.81 IDO1 (0.52) GID4IDO1HTR2BPOLBPKM
SCHEMBL6753945 0.79 TRPC3 (0.55) GID4HTR2BPOLBPKMMAPT
Ammonia Solution, Strong SCHEMBL5028354 0.78 TRPC3 (0.54) GID4HTR2BPOLBPKMMAPT
SCHEMBL2640300 0.78 PARP1 (0.56) GID4HTR2BPOLBPKMMAPT
SCHEMBL10539462 0.77 HTR2B (0.51) GID4IDO1HTR2BPOLBMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0268148-B1 TETRAHYDRONAPHTHALENE DERIVATIVES AND MEDICAMENTS CONTAINING THEM F. HOFFMANN-LA ROCHE AG (CH) 1991-12-11 EP disclosed
US-4808605-A Tetrahydronaphthalene derivatives as calcium antagonists HOFFMANN-LA ROCHE INC. (US) 1989-02-28 US disclosed
EP-0268148-A1 Tetrahydronaphthalene derivatives and medicaments containing them F. HOFFMANN-LA ROCHE AG (CH) 1988-05-25 EP disclosed