SCHEMBL7266507

SCHEMBL7266507

CN1CCC(c2nc(-c3cn(C)c4ccccc34)no2)CC1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 1)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7268767 0.86 HSD11B1 (0.50) ALDH1A1
SCHEMBL7329287 0.86 ALDH1A1 (0.51) ALDH1A1
SCHEMBL7443611 0.86 KCNH2 (0.52) ALDH1A1
Iodide SCHEMBL7266858 0.85 ALDH1A1 (0.50) ALDH1A1
SCHEMBL7268323 0.85 ALDH1A1 (0.52) ALDH1A1
Oxalic Acid SCHEMBL7273813 0.82 HSD11B1 (0.55)
SCHEMBL7327600 0.81 ALDH1A1 (0.48) ALDH1A1
SCHEMBL7267110 0.81 HCRTR1 (0.50) ALDH1A1
SCHEMBL7268778 0.81
Iodide SCHEMBL7266617 0.80 ALDH1A1 (0.47) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0328200-B1 Five-membered ring systems with bonded azacyclic ring substituents MERCK SHARP & DOHME (GB) 1993-12-08 EP claimed
EP-0328200-A1 Five-membered ring systems with bonded azacyclic ring substituents MERCK SHARP & DOHME LTD. (GB) 1989-08-16 EP claimed
EP-0328200-B1 Five-membered ring systems with bonded azacyclic ring substituents MERCK SHARP & DOHME (GB) 1993-12-08 EP disclosed
US-5041456-A Pharmaceutically useful 3-(indol-3-yl)-1,2,4-oxa- and thiadiazoles substituted in the 5-position by an amino containing group MERCK SHARP & DOHME LTD. (GB) 1991-08-20 US disclosed
US-4952587-A PSYCHOLOGICAL DISORDERS, MIGRAINES, ALZHEIMER*S MERCK SHARP & DOHME LTD. (GB) 1990-08-28 US disclosed
EP-0328200-A1 Five-membered ring systems with bonded azacyclic ring substituents MERCK SHARP & DOHME LTD. (GB) 1989-08-16 EP disclosed