SCHEMBL7266703

SCHEMBL7266703

CC1(C)CN(C(=O)NC2CN3CCC2CC3)c2ccccc21

nearest known ligand 0.57

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CHRM2 P08172 2/20 0.53
CHRM1 P11229 2/20 0.53
CHRM3 P20309 2/20 0.53
CHRNA7 P36544 1/20 0.52
NOTUM Q6P988 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7439036 0.99 CHRM2 (0.52) CHRM2CHRM1CHRM3CHRNA7NOTUM
SCHEMBL9602968 0.81 CHRM2 (0.50) CHRM2CHRM1CHRM3CHRNA7
SCHEMBL7265735 0.76 NPC1 (0.61) CHRM2CHRM1CHRM3CHRNA7
Hydrochloric Acid SCHEMBL7446453 0.75 NPC1 (0.60) CHRM2CHRM1CHRM3CHRNA7
Ricasetron SCHEMBL634826 0.73 NOTUM (0.52) NOTUM
Ricasetron SCHEMBL21715163 0.73 NOTUM (0.52) NOTUM
Ricasetron SCHEMBL634827 0.73 NOTUM (0.52) NOTUM
Ricasetron SCHEMBL20362251 0.73 NOTUM (0.52) NOTUM
Ricasetron SCHEMBL7445859 0.72 NOTUM (0.51) NOTUM
SCHEMBL26691209 0.71 NOTUM (0.73) NOTUM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0278173-B1 Use of heterocyclic derivatives in the treatment of depressions GLAXO GROUP LTD (GB) 1993-11-03 EP claimed
EP-0247266-B1 INDOLE DERIVATIVES HAVING AN AZABICYCLIC SIDE CHAIN, PROCESS FOR THEIR PREPARATION, INTERMEDIATES, AND PHARMACEUTICAL COMPOSITIONS BEECHAM GROUP PLC (GB) 1993-03-10 EP claimed
US-5049556-A Certain N-azabicyclo-2,3-dihydro-indole-1-carboxamides having anti-emetic properties, further found useful in treating headaches, neuralgia and anxiety BEECHAM GROUP P.L.C. (GB) 1991-09-17 US claimed
EP-0247266-A1 Indole derivatives having an azabicyclic side chain, process for their preparation, intermediates, and pharmaceutical compositions BEECHAM GROUP PLC (GB) 1987-12-02 EP claimed
EP-0278173-B1 Use of heterocyclic derivatives in the treatment of depressions GLAXO GROUP LTD (GB) 1993-11-03 EP disclosed