Ricasetron

Ricasetron

SCHEMBL634826

CN1[C@@H]2CC[C@H]1C[C@@H](NC(=O)N1CC(C)(C)c3ccccc31)C2

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 1/20 0.52
CNR2 P34972 1/20 0.50
TMEM97 Q5BJF2 1/20 0.47
SIGMAR1 Q99720 1/20 0.47
HTR3A P46098 1/20 0.47
HTR4 Q13639 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Ricasetron SCHEMBL21715163 1.00 NOTUM (0.52) NOTUMCNR2TMEM97SIGMAR1HTR3A
Ricasetron SCHEMBL20362251 1.00 NOTUM (0.52) NOTUMCNR2TMEM97SIGMAR1HTR3A
Ricasetron SCHEMBL634827 1.00 NOTUM (0.52) NOTUMCNR2TMEM97SIGMAR1HTR3A
Ricasetron SCHEMBL7445859 0.99 NOTUM (0.51) NOTUMCNR2TMEM97SIGMAR1HTR3A
SCHEMBL7295216 0.91 NOTUM (0.50) NOTUMCNR2HTR3A
SCHEMBL9368172 0.82 TMEM97 (0.45) TMEM97SIGMAR1HTR3AHTR4
SCHEMBL9602391 0.81 MEN1 (0.42) NOTUM
SCHEMBL7624884 0.81 CNR2 (0.48) NOTUMCNR2HTR3A
SCHEMBL7624888 0.81 CNR2 (0.48) NOTUMCNR2HTR3A
Ethane SCHEMBL7627590 0.80 CNR2 (0.47) NOTUMCNR2HTR3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 405 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20240366639-A1 HETEROCYCLIC GLP-1 AGONISTS GASHERBRUM BIO INC (US) 2024-11-07 US claimed
WO-2023016546-A1 HETEROCYCLIC GLP-1 AGONISTS GASHERBRUM BIO, INC. (US) 2023-02-16 WO claimed
US-11547700-B2 Compositions and methods for treating synucleinopathies CHASE THERAPEUTICS CORPORATION (US) 2023-01-10 US claimed
US-20220146492-A1 CELL MEMBRANE PERMEABILITY RESTORING THERAPY SHINE IAN BASIL (US) 2022-05-12 US claimed
EP-3953000-A1 CELL MEMBRANE PERMEABILITY RESTORING THERAPY Shine, Ian Basil (US) 2022-02-16 EP claimed
WO-2020210643-A1 CELL MEMBRANE PERMEABILITY RESTORING THERAPY SHINE IAN BASIL (US) 2020-10-15 WO claimed
EP-3691637-A1 ORAL BENDAMUSTINE FORMULATIONS TUBE Pharmaceuticals GmbH (AT) 2020-08-12 EP claimed
US-20200246312-A1 ORAL BENDAMUSTINE FORMULATIONS TUBE PHARMACEUTICALS GMBH (AT) 2020-08-06 US claimed
WO-2019068904-A1 ORAL BENDAMUSTINE FORMULATIONS TUBE PHARMACEUTICALS GMBH (AT) 2019-04-11 WO claimed
WO-2016118540-A1 TREATING AND/OR PREVENTING EMESIS AND/OR NAUSEA INCLUDING ACUTE AND/OR DELAYED NAUSEA AND/OR EMESIS Xoc Pharmaceuticals, Inc. (US) 2016-07-28 WO claimed
US-20050209293-A1 Method of treating or inhibiting a non-digestive tract derived abdominal disorder associated with pain using a 5-HT, receptor antagonist SOLVAY PHARMACEUTICALS GMBH (DE) 2005-09-22 US claimed
WO-2005074931-A1 PHARMACEUTICAL COMBINATIONS COMPRISING (S) -PANTOPRAZOLE ALTANA PHARMA AG (DE) 2005-08-18 WO claimed
WO-2004105795-A1 PHARMACEUTICAL COMBINATIONS OF A PROTON PUMP INHIBITOR AND A COMPOUND WHICH MODIFIES GASTROINTESTINAL MOTILITY ALTANA PHARMA AG (DE) 2004-12-09 WO claimed
WO-2003100091-A1 MEANS AND METHODS FOR IMPROVED TREATMENT USING 'SETRONES' EPIDAUROS BIOTECHNOLOGIE AG (DE) 2003-12-04 WO claimed
EP-1336602-A1 Nitrate prodrugs able to release nitric oxide in a controlled and selective way and their use for prevention and treatment of inflammatory, ischemic and proliferative diseases Scaramuzzino, Giovanni (IT) 2003-08-20 EP claimed
WO-2002036113-A1 COMPOSITION COMPRISING: SEROTONIN RECEPTOR ANTAGONISTS (5HT-2, 5HT-3) AND AGONIST (5HT-4) RESPIRATORIUS AB (SE) 2002-05-10 WO claimed
WO-2002036114-A1 COMPOSITION COMPRISING SEROTONIN RECEPTOR ANTAGONISTS, 5 HT-2 AND 5 HT-3 RESPIRATORIUS AB (SE) 2002-05-10 WO claimed
WO-2001095902-A9 A COMPOSITION COMPRISING A COMBINATION OF RECEPTOR AGONISTS AND ANTAGONISTS 2002-04-25 WO claimed
WO-2001095902-A1 A COMPOSITION COMPRISING A COMBINATION OF RECEPTOR AGONISTS AND ANTAGONISTS RESPIRATORIUS AB (SE) 2001-12-20 WO claimed
WO-2001095903-A1 5-HT3 RECEPTOR ANTAGONISTS FOR TREATMENT OF DISORDERS INVOLVING AIRWAY CONSTRICTION RESPIRATORIUS AB (SE) 2001-12-20 WO claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240366639-A1 HETEROCYCLIC GLP-1 AGONISTS GLP1R, GIPR, GCGR NOTUM 3195/4885CNR2 834/4885TMEM97 1320/4885
US-20200246312-A1 ORAL BENDAMUSTINE FORMULATIONS ABCB1, MTHFD1, BHMT NOTUM 987/4885CNR2 914/4885TMEM97 340/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.