SCHEMBL7267407

SCHEMBL7267407

CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@@H](CC(N)=O)C(=O)O

nearest known ligand 0.70

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
PSMB1 P20618 1/20 0.70
CTSK P43235 7/20 0.67
CAPN1 P07384 2/20 0.64
CTSL P07711 3/20 0.64
CTSB P07858 3/20 0.64
CTSS P25774 2/20 0.64

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27429302 0.91 PSMB1 (0.67) PSMB1CTSKCAPN1CTSLCTSB
SCHEMBL27533999 0.91 CTSK (0.70) CTSKCAPN1CTSLCTSBCTSS
SCHEMBL4424261 0.91 CTSK (0.70) CTSKCAPN1CTSLCTSBCTSS
SCHEMBL25406813 0.91 CTSK (0.77) CTSKCAPN1CTSLCTSBCTSS
SCHEMBL20770085 0.91 CTSK (0.77) CTSKCAPN1CTSLCTSBCTSS
SCHEMBL2930262 0.91 CTSK (0.77) CTSKCAPN1CTSLCTSBCTSS
SCHEMBL8823918 0.91 CTSK (0.77) CTSKCAPN1CTSLCTSBCTSS
SCHEMBL4872585 0.91 CTSK (0.77) CTSKCAPN1CTSLCTSBCTSS
SCHEMBL11124167 0.91 MME (0.64) PSMB1CTSKCTSLCTSBCTSS
SCHEMBL14148467 0.91 CTSK (0.77) CTSKCAPN1CTSLCTSBCTSS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5652369-A PROTEASE INHIBITOR HOFFMANN-LA ROCHE INC. (US) 1997-07-29 US disclosed
US-5620987-A Amino acid derivatives HOFFMANN-LA ROCHE INC. (US) 1997-04-15 US disclosed
US-5554756-A PROTEASE INHIBITOR HOFFMANN-LA ROCHE INC. (US) 1996-09-10 US disclosed
US-5446161-A Protease inhibitor, viricides HOFFMANN-LA ROCHE INC. (US) 1995-08-29 US disclosed
EP-0346847-B1 Amino acid derivatives HOFFMANN LA ROCHE (CH) 1994-05-11 EP disclosed
US-5157041-A Viricides HOFFMANN-LA ROCHE INC. (US) 1992-10-20 US disclosed
EP-0346847-A2 Amino acid derivatives F. HOFFMANN-LA ROCHE AG (CH) 1989-12-20 EP disclosed