SCHEMBL7267809

SCHEMBL7267809

COc1cc2nc(-c3ccc(Cl)cc3)nc(N3CCN(CC(=O)N4CCOCC4)CC3)c2cc1OC

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.56
HPGD P15428 1/20 0.56
HIF1A Q16665 1/20 0.56
PIK3CD O00329 2/20 0.54
PIK3R1 P27986 2/20 0.54
PIK3CA P42336 2/20 0.54
PIK3CB P42338 2/20 0.54
PIK3CG P48736 2/20 0.54
PIK3R5 Q8WYR1 2/20 0.54
AURKA O14965 1/20 0.53
SMN1; SMN2 Q16637 1/20 0.51
KDM4E B2RXH2 1/20 0.49
STAT6 P42226 1/20 0.49
NPSR1 Q6W5P4 1/20 0.49
NTSR1 P30989 6/20 0.48
TLR9 Q9NR96 1/20 0.47
L3MBTL1 Q9Y468 1/20 0.47
ACHE P22303 1/20 0.46
BACE1 P56817 1/20 0.46
POLB P06746 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7268671 0.88 AURKA (0.45) ALDH1A1HPGDHIF1APIK3CDPIK3R1
SCHEMBL7267813 0.85 ALDH1A1 (0.70) ALDH1A1HPGDHIF1APIK3CDPIK3R1
SCHEMBL7267791 0.82 NPSR1 (0.52) ALDH1A1HPGDHIF1APIK3CDPIK3R1
SCHEMBL7261541 0.81 KDM4E (0.57) ALDH1A1HPGDHIF1APIK3CDPIK3R1
SCHEMBL13675866 0.78 L3MBTL1 (0.51) ALDH1A1HPGDHIF1APIK3CDPIK3R1
Hydrochloric Acid SCHEMBL7268677 0.77 KDM4E (0.64) ALDH1A1HPGDAURKAKDM4ESTAT6
Hydrochloric Acid SCHEMBL7266340 0.77 SMN1; SMN2 (0.67) ALDH1A1HPGDHIF1ASMN1; SMN2KDM4E
SCHEMBL7262669 0.77 KDM4E (0.76) ALDH1A1HPGDHIF1APIK3CDPIK3R1
SCHEMBL23242448 0.76 ALDH1A1 (0.63) ALDH1A1HPGDHIF1APIK3CDPIK3R1
SCHEMBL7268618 0.76 ALDH1A1 (0.72) ALDH1A1HPGDHIF1APIK3CDPIK3R1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6613772-B1 Drugs such as 2-(p-chlorophenyl-4-(4-hydroxybutyl)amino-6,7,8 -trimethoxyquinazoline used for activation of guanylate cyclase and modulation of cyclic guanosine monophosphate AVENTIS PHARMA DEUTSCHLAND GMBH (DE) 2003-09-02 US disclosed