SCHEMBL7268570

SCHEMBL7268570

COc1cc2nc(-c3ccc(Cl)cc3)nc(N3CC[S+]([O-])CC3)c2cc1OC

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.60
STAT6 P42226 1/20 0.60
NPSR1 Q6W5P4 1/20 0.60
NTSR1 P30989 8/20 0.56
ALDH1A1 P00352 2/20 0.52
HPGD P15428 2/20 0.52
HIF1A Q16665 1/20 0.52
SMN1; SMN2 Q16637 3/20 0.50
HTT P42858 1/20 0.46
ACHE P22303 1/20 0.45
BACE1 P56817 1/20 0.45
PIK3CD O00329 1/20 0.45
PIK3R1 P27986 1/20 0.45
PIK3CA P42336 1/20 0.45
PIK3CB P42338 1/20 0.45
PIK3CG P48736 1/20 0.45
PIK3R5 Q8WYR1 1/20 0.45
GBA1 P04062 1/20 0.43
LMNA P02545 1/20 0.43
TP53 P04637 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7268567 0.90 KDM4E (0.61) KDM4ESTAT6NPSR1NTSR1ALDH1A1
SCHEMBL7262669 0.86 KDM4E (0.76) KDM4ESTAT6NPSR1NTSR1ALDH1A1
SCHEMBL7267789 0.85 KDM4E (0.43) KDM4ESTAT6NPSR1NTSR1ALDH1A1
Hydrochloric Acid SCHEMBL7266340 0.84 SMN1; SMN2 (0.67) KDM4ESTAT6NPSR1NTSR1ALDH1A1
SCHEMBL7267753 0.84 NPSR1 (0.63) KDM4ESTAT6NPSR1NTSR1ALDH1A1
SCHEMBL7267813 0.84 ALDH1A1 (0.70) KDM4ESTAT6NPSR1NTSR1ALDH1A1
SCHEMBL7261541 0.80 KDM4E (0.57) KDM4ESTAT6NPSR1NTSR1ALDH1A1
Hydrochloric Acid SCHEMBL7268677 0.79 KDM4E (0.64) KDM4ESTAT6NPSR1NTSR1ALDH1A1
SCHEMBL7261513 0.79 TSHR (0.57) KDM4ESTAT6NPSR1NTSR1ALDH1A1
SCHEMBL7261387 0.78 KDM4E (0.71) KDM4ESTAT6NPSR1NTSR1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6613772-B1 Drugs such as 2-(p-chlorophenyl-4-(4-hydroxybutyl)amino-6,7,8 -trimethoxyquinazoline used for activation of guanylate cyclase and modulation of cyclic guanosine monophosphate AVENTIS PHARMA DEUTSCHLAND GMBH (DE) 2003-09-02 US disclosed
EP-1040101-A1 SUBSTITUTED 2-ARYL-4-AMINO-CHINAZOLINES, METHOD FOR THE PRODUCTION AND USE THEREOF AS MEDICAMENTS Aventis Pharma Deutschland GmbH (DE) 2000-10-04 EP disclosed
WO-1999032460-A1 SUBSTITUTED 2-ARYL-4-AMINO-CHINAZOLINES, METHOD FOR THE PRODUCTION AND USE THEREOF AS MEDICAMENTS AVENTIS PHARMA DEUTSCHLAND GMBH (DE) 1999-07-01 WO disclosed