SCHEMBL7267753

SCHEMBL7267753

COc1cc2nc(-c3ccc(Cl)cc3)nc(N3CCSCC3)c2cc1OC

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 3/20 0.63
KDM4E B2RXH2 2/20 0.63
STAT6 P42226 1/20 0.63
NTSR1 P30989 8/20 0.58
ALDH1A1 P00352 3/20 0.53
HPGD P15428 2/20 0.53
HIF1A Q16665 1/20 0.53
SMN1; SMN2 Q16637 3/20 0.52
CYP1A2 P05177 2/20 0.48
CYP2C9 P11712 2/20 0.48
CYP2C19 P33261 2/20 0.48
POLB P06746 1/20 0.48
HTT P42858 1/20 0.47
ACHE P22303 1/20 0.47
BACE1 P56817 1/20 0.47
PIK3CD O00329 1/20 0.46
PIK3R1 P27986 1/20 0.46
PIK3CA P42336 1/20 0.46
PIK3CB P42338 1/20 0.46
PIK3CG P48736 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7266516 0.90 KDM4E (0.64) NPSR1KDM4ESTAT6NTSR1ALDH1A1
SCHEMBL7262669 0.88 KDM4E (0.76) NPSR1KDM4ESTAT6NTSR1ALDH1A1
SCHEMBL7267813 0.86 ALDH1A1 (0.70) NPSR1KDM4ESTAT6NTSR1ALDH1A1
Hydrochloric Acid SCHEMBL7266340 0.86 SMN1; SMN2 (0.67) NPSR1KDM4ESTAT6NTSR1ALDH1A1
SCHEMBL7261986 0.84 NPSR1 (0.47) NPSR1KDM4ESTAT6NTSR1ALDH1A1
SCHEMBL7268570 0.84 KDM4E (0.60) NPSR1KDM4ESTAT6NTSR1ALDH1A1
SCHEMBL4091890 0.83 NPSR1 (0.57) NPSR1KDM4ESTAT6ALDH1A1SMN1; SMN2
SCHEMBL7261541 0.82 KDM4E (0.57) NPSR1KDM4ESTAT6NTSR1ALDH1A1
Hydrochloric Acid SCHEMBL7268677 0.80 KDM4E (0.64) NPSR1KDM4ESTAT6NTSR1ALDH1A1
SCHEMBL7261513 0.80 TSHR (0.57) NPSR1KDM4ESTAT6NTSR1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6613772-B1 Drugs such as 2-(p-chlorophenyl-4-(4-hydroxybutyl)amino-6,7,8 -trimethoxyquinazoline used for activation of guanylate cyclase and modulation of cyclic guanosine monophosphate AVENTIS PHARMA DEUTSCHLAND GMBH (DE) 2003-09-02 US disclosed
EP-1040101-A1 SUBSTITUTED 2-ARYL-4-AMINO-CHINAZOLINES, METHOD FOR THE PRODUCTION AND USE THEREOF AS MEDICAMENTS Aventis Pharma Deutschland GmbH (DE) 2000-10-04 EP disclosed
WO-1999032460-A1 SUBSTITUTED 2-ARYL-4-AMINO-CHINAZOLINES, METHOD FOR THE PRODUCTION AND USE THEREOF AS MEDICAMENTS AVENTIS PHARMA DEUTSCHLAND GMBH (DE) 1999-07-01 WO disclosed