SCHEMBL7269135

SCHEMBL7269135

c1ccc(CCC2(CCc3ccccc3)CO2)cc1

nearest known ligand 0.46

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 2/20 0.43
MAOA P21397 2/20 0.43
MAOB P27338 2/20 0.43
ALDH1A1 P00352 2/20 0.42
HPGD P15428 1/20 0.42
ALOX15 P16050 1/20 0.42
ALOX12 P18054 1/20 0.42
CASP1 P29466 1/20 0.42
HSD17B10 Q99714 1/20 0.42
TDP1 Q9NUW8 2/20 0.41
CYP2A6 P11509 1/20 0.41
HTR2A P28223 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
TAAR1 Q96RJ0 1/20 0.41
LOXL2 Q9Y4K0 1/20 0.41
KCNH2 Q12809 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12144581 0.89 KDM1A (0.48) KDM1AMAOAMAOBTDP1HTR2A
SCHEMBL6957893 0.88 TDP1 (0.45) KDM1AMAOAMAOBALDH1A1TDP1
SCHEMBL7270639 0.86 KDM1A (0.38) KDM1AMAOAMAOBALDH1A1HPGD
SCHEMBL7404874 0.82 TSHR (0.45) KDM1AMAOAMAOBTDP1TAAR1
SCHEMBL1376365 0.78 TAAR1 (0.45) KDM1AALDH1A1CYP2A6HTR2ATAAR1
SCHEMBL22013858 0.78 GAA (0.41) KDM1AMAOAMAOBALDH1A1HPGD
SCHEMBL13082818 0.78 OPRM1 (0.44) KDM1AMAOAMAOBALDH1A1HPGD
SCHEMBL7997821 0.78 GAA (0.41) KDM1AMAOAMAOBALDH1A1HPGD
SCHEMBL11825227 0.77 OPRM1 (0.42) KDM1AMAOAMAOBALDH1A1HPGD
SCHEMBL23611125 0.76 MAOA (0.48) KDM1AMAOAMAOBALDH1A1LOXL2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0839798-A2 Intermediates for preparating non-peptide retroviral protease inhibitors ABBOTT LABORATORIES (US) 1998-05-06 EP disclosed
US-5670675-A Retroviral protease inhibiting compounds ABBOTT LABORATORIES (US) 1997-09-23 US disclosed
US-5545750-A TREATING HUMAN IMMUNODEFICIENCY VIRUS ABBOTT LABORATORIES (US) 1996-08-13 US disclosed
US-5142056-A Human immunodeficiency virus protease inhibitor ABBOTT LABORATORIES (US) 1992-08-25 US disclosed
EP-0402646-A1 Retroviral protease inhibiting compounds ABBOTT LABORATORIES (US) 1990-12-19 EP disclosed