SCHEMBL7269223

SCHEMBL7269223

[CH2]CCCNC(=O)c1ccc(C(=O)O)cc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 1/20 0.56
ALDH1A1 P00352 1/20 0.53
NPC1 O15118 4/20 0.50
RAB9A P51151 4/20 0.50
NAAA Q02083 1/20 0.49
HDAC3 O15379 1/20 0.49
HDAC4 P56524 1/20 0.49
HDAC1 Q13547 1/20 0.49
HDAC7 Q8WUI4 1/20 0.49
HDAC2 Q92769 1/20 0.49
HDAC10 Q969S8 1/20 0.49
HDAC11 Q96DB2 1/20 0.49
HDAC8 Q9BY41 1/20 0.49
HDAC6 Q9UBN7 1/20 0.49
HDAC9 Q9UKV0 1/20 0.49
HDAC5 Q9UQL6 1/20 0.49
L3MBTL1 Q9Y468 1/20 0.47
LMNA P02545 1/20 0.47
POLB P06746 1/20 0.47
HSP90AA1 P07900 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1014753 0.87 NPC1 (0.66) MAPK1NPC1RAB9ANAAAHDAC3
SCHEMBL10363539 0.86 MAPK1 (0.72) MAPK1ALDH1A1NPC1RAB9ANAAA
SCHEMBL5612077 0.84 DRD2 (0.64) NPC1RAB9AHDAC3HDAC4HDAC1
SCHEMBL10173739 0.81 NAAA (0.67) MAPK1ALDH1A1NPC1RAB9ANAAA
SCHEMBL16557239 0.81 POLB (0.68) MAPK1ALDH1A1NPC1RAB9ANAAA
SCHEMBL1556347 0.81 HDAC1 (0.67) MAPK1ALDH1A1NPC1RAB9ANAAA
SCHEMBL27447913 0.81 EPHX2 (0.49) MAPK1ALDH1A1NPC1RAB9AHDAC1
SCHEMBL8353635 0.80 MAPK1 (0.59) MAPK1ALDH1A1NPC1RAB9ANAAA
SCHEMBL5097388 0.80 NAAA (0.66) ALDH1A1NPC1RAB9ANAAAHDAC2
SCHEMBL1416823 0.80 HDAC1 (0.70) MAPK1ALDH1A1NPC1RAB9ANAAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0236872-B1 HYDROXYL AMINE DERIVATIVES, THEIR PREPARATION AND USE AS MEDICAMENTS F. HOFFMANN-LA ROCHE AG (CH) 1992-11-25 EP claimed
US-4996358-A Control, prevention rheumatic diseases HOFFMANN-LA ROCHE INC. (US) 1991-02-26 US claimed
EP-0236872-A2 Hydroxyl amine derivatives, their preparation and use as medicaments F. HOFFMANN-LA ROCHE AG (CH) 1987-09-16 EP claimed
EP-0236872-B1 HYDROXYL AMINE DERIVATIVES, THEIR PREPARATION AND USE AS MEDICAMENTS F. HOFFMANN-LA ROCHE AG (CH) 1992-11-25 EP disclosed
EP-0423943-A2 Use of collagenase inhibitors in the treatment of demyelinating diseases, in particular multiple sclerosis Beecham Group p.l.c. (GB) 1991-04-24 EP disclosed
US-4996358-A Control, prevention rheumatic diseases HOFFMANN-LA ROCHE INC. (US) 1991-02-26 US disclosed
EP-0236872-A2 Hydroxyl amine derivatives, their preparation and use as medicaments F. HOFFMANN-LA ROCHE AG (CH) 1987-09-16 EP disclosed