SCHEMBL7270034

SCHEMBL7270034

CC(C)C(NC(=O)N1CCN(C)CC1)C(=O)O.[LiH]

nearest known ligand 0.44

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.42
ALDH1A1 P00352 4/20 0.42
KDM4C Q9H3R0 1/20 0.42
CYP2C19 P33261 1/20 0.40
CYP1A2 P05177 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
PKM P14618 1/20 0.39
EPHX2 P34913 2/20 0.38
POLB P06746 2/20 0.37
HTR1A P08908 1/20 0.37
GAA P10253 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6447920 0.98 KDM4E (0.43) KDM4EALDH1A1KDM4CCYP2C19CYP1A2
SCHEMBL5711205 0.98 KDM4E (0.43) KDM4EALDH1A1KDM4CCYP2C19CYP1A2
Lithium SCHEMBL7270041 0.97 KDM4E (0.42) KDM4EALDH1A1KDM4CCYP2C19CYP1A2
SCHEMBL7339063 0.82 SMN1; SMN2 (0.45) ALDH1A1CYP2C19CYP1A2SMN1; SMN2MEN1
SCHEMBL7339055 0.82 SMN1; SMN2 (0.45) ALDH1A1CYP2C19CYP1A2SMN1; SMN2MEN1
SCHEMBL7308065 0.81 MEN1 (0.52) KDM4EALDH1A1KDM4CCYP1A2TDP1
SCHEMBL7279963 0.81 MEN1 (0.52) KDM4EALDH1A1KDM4CCYP1A2TDP1
Lithium Ion SCHEMBL7270031 0.81 CYP1A2 (0.38) KDM4EALDH1A1KDM4CCYP2C19CYP1A2
SCHEMBL6447284 0.81 RAB9A (0.49) ALDH1A1CYP1A2SMN1; SMN2MEN1KMT2A
SCHEMBL6447936 0.81 RAB9A (0.49) ALDH1A1CYP1A2SMN1; SMN2MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0839798-A2 Intermediates for preparating non-peptide retroviral protease inhibitors ABBOTT LABORATORIES (US) 1998-05-06 EP disclosed
US-5670675-A Retroviral protease inhibiting compounds ABBOTT LABORATORIES (US) 1997-09-23 US disclosed
US-5545750-A TREATING HUMAN IMMUNODEFICIENCY VIRUS ABBOTT LABORATORIES (US) 1996-08-13 US disclosed
US-5142056-A Human immunodeficiency virus protease inhibitor ABBOTT LABORATORIES (US) 1992-08-25 US disclosed
EP-0402646-A1 Retroviral protease inhibiting compounds ABBOTT LABORATORIES (US) 1990-12-19 EP disclosed