SCHEMBL7270417

SCHEMBL7270417

COC1CN[C@H](C(=O)OC(C)(C)C)C1

nearest known ligand 0.36

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CTSC P53634 1/20 0.36
MAPK1 P28482 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.30
CHRM2 P08172 1/20 0.30
CHRM1 P11229 1/20 0.30
CHRM3 P20309 1/20 0.30
CHRNB2 P17787 1/20 0.30
CHRNB4 P30926 1/20 0.30
CHRNA3 P32297 1/20 0.30
CHRNA7 P36544 1/20 0.30
CHRNA4 P43681 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25930148 1.00 CTSC (0.36) CTSCMAPK1L3MBTL1CHRM2CHRM1
SCHEMBL594328 0.86 MAPK1 (0.31) MAPK1L3MBTL1CHRM2CHRM1CHRM3
SCHEMBL11449860 0.86 MAPK1 (0.31) MAPK1L3MBTL1CHRM2CHRM1CHRM3
SCHEMBL11449155 0.85 HRH3 (0.31) MAPK1
Hydrochloric Acid SCHEMBL29398060 0.85 MAPK1 (0.30) MAPK1
SCHEMBL11467239 0.82 NFKB1 (0.30)
SCHEMBL6199839 0.82 CTSC (0.42) CTSCCHRNB2CHRNB4CHRNA3CHRNA7
SCHEMBL11449583 0.82 CTSC (0.42) CTSCCHRNB2CHRNB4CHRNA3CHRNA7
SCHEMBL7021231 0.82 CTSC (0.42) CTSCCHRNB2CHRNB4CHRNA3CHRNA7
SCHEMBL3834619 0.82 CTSC (0.42) CTSCCHRNB2CHRNB4CHRNA3CHRNA7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0048159-A2 Novel carboxyalkyl peptides and thioethers and ethers of peptides as antihypertensive agents UNIVERSITY OF MIAMI (US) 1982-03-24 EP disclosed
US-4221912-A Dithio derivatives of 4,5-dihydro-1H-pyrrole-2-carboxylic acids and 1,4,5,6-tetrahydropyridine-2-carboxylic acids E. R. SQUIBB & SONS, INC. (US) 1980-09-09 US disclosed
US-4217458-A Acylmercaptoacyl derivatives of 4,5-dihydro-1H-pyrrole-2-carboxylic acids and 1,4,5,6-tetrahydropyridine-2-carboxylic acids E. R. SQUIBB & SONS, INC. (US) 1980-08-12 US disclosed
US-4198515-A Mercaptoacyl derivatives of 4,5-dihydro-1H-pyrrole-2-carboxylic acids and 1,4,5,6-tetrahydropyridine-2-carboxylic acids E. R. SQUIBB & SONS, INC. (US) 1980-04-15 US disclosed