SCHEMBL7270906

SCHEMBL7270906

Cc1ccc(-n2c(=O)oc(=O)c3cccnc32)cc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 3/20 0.51
CYP2C19 P33261 2/20 0.51
CYP1A2 P05177 1/20 0.51
CYP2C9 P11712 1/20 0.51
ALDH1A1 P00352 3/20 0.49
KAT2B Q92831 1/20 0.45
AKT1 P31749 1/20 0.44
AKT2 P31751 1/20 0.44
TSHR P16473 2/20 0.44
FEN1 P39748 1/20 0.42
PDE4B Q07343 3/20 0.40
PDE4A P27815 2/20 0.40
PDE4C Q08493 2/20 0.40
PDE4D Q08499 2/20 0.40
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
POLB P06746 1/20 0.40
MAPK1 P28482 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1522773 0.87 FEN1 (0.55) CYP2C19ALDH1A1KAT2BTSHRFEN1
SCHEMBL7278555 0.85 POLB (0.43) HPGDCYP2C19CYP1A2CYP2C9ALDH1A1
SCHEMBL7278394 0.85 LMNA (0.51) ALDH1A1KAT2BPDE4BNPC1RAB9A
SCHEMBL7281964 0.78 HPGD (0.53) HPGDCYP2C19CYP1A2ALDH1A1TSHR
SCHEMBL7281855 0.78 KAT2B (0.50) HPGDCYP1A2ALDH1A1KAT2BPDE4B
SCHEMBL2412984 0.77 KMT2A (0.55) HPGDCYP2C19CYP1A2ALDH1A1TSHR
SCHEMBL1522225 0.77 PTGDR2 (0.55) HPGDALDH1A1KAT2BSMN1; SMN2TP53
SCHEMBL11240235 0.75 FEN1 (0.51) HPGDCYP2C19CYP1A2CYP2C9ALDH1A1
SCHEMBL2409225 0.73 PDE4A (0.57) ALDH1A1KAT2BPDE4BPDE4APDE4C
SCHEMBL11978691 0.73 CYP2C19 (0.49) HPGDCYP2C19CYP1A2CYP2C9ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0459505-B1 Imidazonaphthyridine derivatives KYOWA HAKKO KOGYO KK (JP) 1996-10-02 EP disclosed
US-5536730-A ANTIINFLAMMATORY, ANTIALLERGIC AND BRONCHODILATIVE ACTIVITY KYOWA HAKKO KOGYO CO. LTD. (JP) 1996-07-16 US disclosed
US-5468756-A Antiinflammatory, antiallergen KYOWA HAKKO KOGYO CO., LTD. (JP) 1995-11-21 US disclosed
US-5364859-A Antiinflammatory agents, antiallergens, bronchodilators KYOWA HAKKO KOGYO CO., LTD. (JP) 1994-11-15 US disclosed
EP-0459505-A1 Imidazonaphthyridine derivatives KYOWA HAKKO KOGYO CO., LTD. (JP) 1991-12-04 EP disclosed