SCHEMBL7271102

SCHEMBL7271102

O=Cc1c(F)cc(Cl)cc1C(F)(F)F

nearest known ligand 0.39

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 3/20 0.39
EPAS1 Q99814 3/20 0.33
HTR2A P28223 1/20 0.33
HTR2C P28335 1/20 0.33
ERN1 O75460 1/20 0.32
CYP2D6 P10635 2/20 0.32
CYP2C9 P11712 1/20 0.32
CYP1A2 P05177 1/20 0.32
CYP2C19 P33261 1/20 0.32
RAB9A P51151 1/20 0.32
AHR P35869 1/20 0.31
HSD11B1 P28845 1/20 0.31
SLC22A12 Q96S37 2/20 0.30
MEN1 O00255 1/20 0.30
ALDH1A1 P00352 1/20 0.30
KMT2A Q03164 1/20 0.30
TDP1 Q9NUW8 1/20 0.30
DDR1 Q08345 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1349783 0.81 ERN1 (0.41) EPAS1ERN1CYP2C9CYP2C19MEN1
SCHEMBL9342725 0.80 KIF11 (0.41) KIF11ERN1CYP2D6CYP2C9
SCHEMBL22620620 0.79 RAB9A (0.32) KIF11EPAS1ERN1CYP2D6CYP1A2
SCHEMBL424780 0.78 KIF11 (0.40) KIF11CYP2D6CYP2C9MEN1KMT2A
SCHEMBL9342595 0.76 KIF11 (0.38) KIF11EPAS1CYP2D6CYP2C9
SCHEMBL6060504 0.75 ERN1 (0.42) ERN1MEN1ALDH1A1KMT2ATDP1
SCHEMBL7926449 0.73 KIF11 (0.42) KIF11EPAS1CYP2D6CYP2C9MEN1
SCHEMBL29560171 0.73 KIF11 (0.35) KIF11EPAS1HSD11B1MEN1ALDH1A1
SCHEMBL9340556 0.73 KIF11 (0.35) KIF11EPAS1HSD11B1MEN1ALDH1A1
SCHEMBL18795660 0.73 ERN1 (0.45) KIF11EPAS1HTR2AHTR2CERN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0396987-A2 Nuclear fluorinated trifluoromethylbenzaldehydes BAYER AG (DE) 1990-11-14 EP claimed
US-5041683-A Nuclear-fluorinated trifluoromethylbenzaldehydes BAYER AKTIENGESELLSCHAFT (DE) 1991-08-20 US disclosed
EP-0396987-A2 Nuclear fluorinated trifluoromethylbenzaldehydes BAYER AG (DE) 1990-11-14 EP disclosed
EP-0174131-A2 Dihydropyridines, processes and intermediates for their production, and pharmaceutical formulations containing them FISONS plc (GB) 1986-03-12 EP disclosed