SCHEMBL7272071

SCHEMBL7272071

Nc1nc(S)c2ncn(C[C@H](N)C(=O)O)c2n1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCNE1 P24864 4/20 0.43
CDK2 P24941 4/20 0.43
ALDH1A1 P00352 2/20 0.43
CYP2C19 P33261 2/20 0.41
HDAC6 Q9UBN7 6/20 0.40
HDAC1 Q13547 5/20 0.40
CDK1 P06493 3/20 0.40
CCNB1 P14635 3/20 0.40
HDAC4 P56524 1/20 0.40
SLC29A1 Q99808 1/20 0.40
CYP1A2 P05177 2/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2C9 P11712 1/20 0.35
HIF1A Q16665 1/20 0.35
PHLPP2 Q6ZVD8 1/20 0.35
ADORA2A P29274 1/20 0.35
ADORA1 P30542 1/20 0.35
HSP90AA1 P07900 1/20 0.34
HSP90AB1 P08238 1/20 0.34
HDAC2 Q92769 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7272082 1.00 CCNE1 (0.43) CCNE1CDK2ALDH1A1CYP2C19HDAC6
SCHEMBL7271581 0.85 CCNE1 (0.44) CCNE1CDK2ALDH1A1CYP2C19HDAC6
SCHEMBL7271567 0.85 CCNE1 (0.44) CCNE1CDK2ALDH1A1CYP2C19HDAC6
SCHEMBL7279752 0.81 ALDH1A1 (0.54) ALDH1A1CYP3A4ADORA2AADORA1
SCHEMBL7279764 0.81 ALDH1A1 (0.54) ALDH1A1CYP3A4ADORA2AADORA1
SCHEMBL9388321 0.81 CYP2C19 (0.47) CCNE1CDK2ALDH1A1CYP2C19HDAC6
SCHEMBL28187282 0.75 PNP (0.58) ALDH1A1CYP3A4HIF1A
SCHEMBL10683911 0.74 ALDH1A1 (0.75) ALDH1A1CYP3A4ADORA2AADORA1
SCHEMBL2270408 0.74 ALDH1A1 (0.75) ALDH1A1CYP3A4ADORA2AADORA1
SCHEMBL7262136 0.72 CYP3A4 (0.64) CCNE1CDK2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4766110-A INHIBITS ANGIOTENSIN CONVERTING ENZYME, HYPOTENSIVE AGENTS RYAN JAMES W (US) 1988-08-23 US disclosed
EP-0073143-B1 NOVEL COMPLEX AMIDO AND IMIDO DERIVATIVES OF CARBOXYALKYL PEPTIDES AND THIOETHERS AND ETHERS OF PEPTIDES Ryan, James Walter (US) 1985-11-21 EP disclosed
EP-0048159-A2 Novel carboxyalkyl peptides and thioethers and ethers of peptides as antihypertensive agents UNIVERSITY OF MIAMI (US) 1982-03-24 EP disclosed