SCHEMBL7272145

SCHEMBL7272145

COc1ccc(-c2nc3cnc(Cl)cc3[nH]2)c(OC)c1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE2A O00408 1/20 0.56
AMY1A P0DUB6 11/20 0.52
RUNX1 Q01196 2/20 0.45
KDM4E B2RXH2 2/20 0.44
NPC1 O15118 2/20 0.44
RAB9A P51151 2/20 0.44
ALDH1A1 P00352 1/20 0.44
TP53 P04637 1/20 0.44
HPGD P15428 1/20 0.44
TSHR P16473 1/20 0.44
NFKB1 P19838 1/20 0.44
NFKB2 Q00653 1/20 0.44
RELA Q04206 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
HSD17B10 Q99714 1/20 0.44
CYP1A2 P05177 1/20 0.44
CYP3A4 P08684 1/20 0.44
PDE5A O76074 1/20 0.43
PDE3B Q13370 1/20 0.43
PDE3A Q14432 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7280668 0.86 PDE2A (0.57) PDE2AAMY1ARUNX1KDM4ENPC1
SCHEMBL7280215 0.83 PDE2A (0.54) PDE2AAMY1ARUNX1KDM4ENPC1
SCHEMBL10734755 0.82 PDE2A (0.57) PDE2AAMY1ARUNX1KDM4ENPC1
SCHEMBL13406023 0.80 AMY1A (0.60) PDE2AAMY1AKDM4ENPC1RAB9A
SCHEMBL7270959 0.80 PDE2A (0.58) PDE2AAMY1AKDM4ENPC1RAB9A
Hydrochloric Acid SCHEMBL7272531 0.79 PDE2A (0.57) PDE2AAMY1AKDM4ENPC1RAB9A
SCHEMBL3337825 0.78 PDE2A (0.66) PDE2AAMY1ARUNX1KDM4ENPC1
SCHEMBL10690574 0.76 PDE2A (0.51) PDE2AAMY1ARUNX1KDM4EALDH1A1
SCHEMBL12470674 0.75 PDE2A (0.56) PDE2AAMY1AKDM4ENPC1RAB9A
SCHEMBL10846574 0.75 PDE2A (0.62) PDE2AAMY1AKDM4EALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4904785-A INOTROPIC AGENTS FOR CARDIOVASCULAR DISORDERS ELI LILLY AND COMPANY (US) 1990-02-27 US disclosed
US-4758574-A 2-phenylimidazio (4,5-c) pyridines ELI LILLY AND COMPANY (US) 1988-07-19 US disclosed
EP-0093593-A2 Pyridine compounds ELI LILLY AND COMPANY (US) 1983-11-09 EP disclosed