SCHEMBL10690574

SCHEMBL10690574

COc1ccc(-c2nc3cnc(OC)nc3[nH]2)c(OC)c1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE2A O00408 1/20 0.51
CYP1A2 P05177 2/20 0.45
CYP3A4 P08684 2/20 0.45
KDM4E B2RXH2 1/20 0.45
ALDH1A1 P00352 1/20 0.42
GAA P10253 1/20 0.42
MAPK1 P28482 1/20 0.42
HTT P42858 1/20 0.42
GFER P55789 1/20 0.42
AMY1A P0DUB6 3/20 0.41
CYP1A1 P04798 2/20 0.40
CYP1B1 Q16678 2/20 0.40
CTSG P08311 1/20 0.40
KLK7 P49862 1/20 0.40
CTRC Q99895 1/20 0.40
KLK14 Q9P0G3 1/20 0.40
KLK5 Q9Y337 1/20 0.40
HDAC3 O15379 1/20 0.39
HDAC4 P56524 1/20 0.39
HDAC1 Q13547 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10686647 0.90 PDE2A (0.42) PDE2ACYP1A2CYP3A4KDM4EALDH1A1
SCHEMBL10610355 0.87 PDE2A (0.40) PDE2ACYP1A2CYP3A4KDM4EGAA
SCHEMBL10689035 0.86 ESR1 (0.42) PDE2AGAAAMY1APDE5APDE3B
SCHEMBL10690513 0.86 AMY1A (0.47) PDE2ACYP1A2CYP3A4ALDH1A1MAPK1
SCHEMBL10685926 0.85 PDGFRB (0.48) PDE2ACYP3A4KDM4EMAPK1CYP2E1
SCHEMBL10691788 0.85 PDE2A (0.46) PDE2ACYP1A2CYP3A4KDM4EALDH1A1
SCHEMBL10690462 0.84 AMY1A (0.40) CYP1A2KDM4EALDH1A1AMY1APDE5A
SCHEMBL10685567 0.84 GUSB (0.54) KDM4EALDH1A1GAAHTTAMY1A
SCHEMBL10691944 0.83 GUSB (0.38) PDE2AKDM4EALDH1A1MAPK1HTT
SCHEMBL11237399 0.82 PDE2A (0.51) PDE2ACYP1A2CYP3A4KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4722929-A Novel 2-phenyl-imidazoles and pharmaceutical compositions containing same DR. KARL THOMAE GMBH (DE) 1988-02-02 US disclosed
EP-0149200-A1 Novel 2-pnenyl-imidazoles, their preparation and drugs containing them Dr. Karl Thomae GmbH (DE) 1985-07-24 EP disclosed