SCHEMBL7272147

SCHEMBL7272147

CCCc1c(C=O)cc([N+](=O)[O-])c(OC)c1OC

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.49
MAPT P10636 3/20 0.49
KDM4E B2RXH2 1/20 0.49
CYP3A4 P08684 1/20 0.49
ALOX15 P16050 1/20 0.49
PRKDC P78527 1/20 0.49
HSD17B10 Q99714 1/20 0.49
ERN1 O75460 5/20 0.38
TPMT P51580 1/20 0.38
ALDH3A1 P30838 2/20 0.38
TUBB4A P04350 1/20 0.36
TUBB P07437 1/20 0.36
TUBA3C P0DPH7 1/20 0.36
TUBA1B P68363 1/20 0.36
TUBA4A P68366 1/20 0.36
TUBB4B P68371 1/20 0.36
TUBB3 Q13509 1/20 0.36
TUBB2A Q13885 1/20 0.36
TUBB8 Q3ZCM7 1/20 0.36
TUBA3E Q6PEY2 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7279701 0.89 KDM4E (0.44) ALDH1A1MAPTKDM4ECYP3A4ALOX15
SCHEMBL7279476 0.88 MAPT (0.42) ALDH1A1MAPTKDM4ECYP3A4ALOX15
SCHEMBL7273865 0.77 TPMT (0.37) ALDH1A1MAPTKDM4ECYP3A4ALOX15
SCHEMBL5653572 0.77 ALDH1A1 (0.53) ALDH1A1MAPTKDM4ECYP3A4ALOX15
SCHEMBL4437002 0.77 ERN1 (0.55) ALDH1A1MAPTKDM4ECYP3A4ALOX15
SCHEMBL7280419 0.76 ALDH1A1 (0.37) ALDH1A1KDM4EPRKDCERN1TUBB1
SCHEMBL22411776 0.74 ALDH1A1 (0.53) ALDH1A1MAPTKDM4ECYP3A4ALOX15
SCHEMBL17113788 0.72 MAPT (0.54) ALDH1A1MAPTKDM4ECYP3A4ALOX15
SCHEMBL31454148 0.72 ERN1 (0.56) ALDH1A1MAPTKDM4ECYP3A4ALOX15
SCHEMBL9550827 0.72 ERN1 (0.52) ALDH1A1MAPTKDM4ECYP3A4ALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4885313-A 3,4-Dihydroxyphenylethylamine derivatives and their use FISONS PLC (GB) 1989-12-05 US disclosed
US-4803225-A Dihydroxy-phenethylamino compounds useful as pharmaceuticals FISONS, PLC (GB) 1989-02-07 US disclosed
US-4720586-A Substituted 3,4-dihydroxy-phenylethylamino compounds FISONS, PLC (GB) 1988-01-19 US disclosed
EP-0142283-A2 Phenylethylamines, process for their preparation and compositions containing them FISONS plc (GB) 1985-05-22 EP disclosed