SCHEMBL7272211

SCHEMBL7272211

C=CC[C@@H]1C[C@@H](COc2ccc(CCCCNC(=O)OC(C)(C)C)cc2)N(CCc2ccc3ccccc3c2)C1=O

nearest known ligand 0.38

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 3/20 0.38
CCNC P24863 1/20 0.35
CDK8 P49336 1/20 0.35
ASAH1 Q13510 1/20 0.35
CA12 O43570 4/20 0.35
CA1 P00915 4/20 0.35
CA2 P00918 4/20 0.35
CA9 Q16790 4/20 0.35
CES2 O00748 1/20 0.34
NAMPT P43490 1/20 0.34
TLR2 O60603 1/20 0.34
TLR1 Q15399 1/20 0.34
DRD2 P14416 3/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7282368 0.93 SIGMAR1 (0.44) SIGMAR1CA12CA1CA2CA9
SCHEMBL7282728 0.91 SIGMAR1 (0.40) SIGMAR1CCNCCDK8ASAH1CA12
SCHEMBL7274358 0.90 SIGMAR1 (0.44) SIGMAR1CA12CA1CA2CA9
SCHEMBL7283476 0.90 SIGMAR1 (0.45) SIGMAR1CA12CA1CA2CA9
SCHEMBL7275605 0.89 NQO2 (0.38) SIGMAR1
SCHEMBL7275258 0.88 CA12 (0.41) SIGMAR1CA12CA1CA2CA9
SCHEMBL7275517 0.88 SIGMAR1 (0.43) SIGMAR1
SCHEMBL7272287 0.87 SIGMAR1 (0.42) SIGMAR1CA12CA1CA2CA9
SCHEMBL7281590 0.87 SIGMAR1 (0.44) SIGMAR1
SCHEMBL7280624 0.86 SIGMAR1 (0.45) SIGMAR1CA1CA2NAMPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5591769-A PYRROLIDINE DERIVATIVES; ANTICOAGULANTS KARL THOMAE GMBH (DE) 1997-01-07 US disclosed
US-5541343-A ANTIAGGLOMERANTS FOR CELLS OR ANTICOAGULANTS KARL THOMAE GMBH (DE) 1996-07-30 US disclosed
EP-0483667-A2 Cyclic imino derivatives, process for their preparation and drugs containing them Dr. Karl Thomae GmbH (DE) 1992-05-06 EP disclosed