SCHEMBL7272269

SCHEMBL7272269

Cn1cc(C#N)c(Nc2ccccc2[N+](=O)[O-])n1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 3/20 0.46
ALDH1A1 P00352 3/20 0.46
TDP1 Q9NUW8 2/20 0.46
L3MBTL1 Q9Y468 2/20 0.46
CASP7 P55210 1/20 0.46
HTT P42858 1/20 0.44
ABCG2 Q9UNQ0 3/20 0.43
EGFR P00533 2/20 0.42
MAPT P10636 6/20 0.42
MEN1 O00255 4/20 0.42
KMT2A Q03164 4/20 0.42
RAB9A P51151 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
GAA P10253 1/20 0.42
PKM P14618 1/20 0.42
LMNA P02545 2/20 0.41
POLB P06746 1/20 0.38
CYP1A2 P05177 1/20 0.38
CCNA2 P20248 1/20 0.38
CDK2 P24941 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7263514 0.84 MAPT (0.45) MAPK1ALDH1A1TDP1L3MBTL1HTT
SCHEMBL7264081 0.83 ALDH3A1 (0.40) MAPK1ALDH1A1TDP1L3MBTL1HTT
SCHEMBL7263524 0.83 VCAM1 (0.52) MAPK1ALDH1A1TDP1L3MBTL1HTT
SCHEMBL7263522 0.83 KDM4E (0.41) MAPK1L3MBTL1HTTEGFRMEN1
SCHEMBL10991410 0.83 HTT (0.38) ALDH1A1L3MBTL1HTTMAPTMEN1
SCHEMBL7263501 0.83 VCAM1 (0.49) MAPK1ALDH1A1TDP1L3MBTL1HTT
SCHEMBL7272454 0.82 POLB (0.38) MAPK1ALDH1A1TDP1HTTMAPT
SCHEMBL7272347 0.80 MAPK1 (0.52) MAPK1ALDH1A1MAPTMEN1KMT2A
SCHEMBL7271277 0.80 MERTK (0.45) ALDH1A1TDP1L3MBTL1HTTMAPT
SCHEMBL11000243 0.80 MAPK1 (0.46) MAPK1ALDH1A1TDP1L3MBTL1CASP7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4542131-A NERVOUS SYSTEM DISORDERS LILLY INDUSTRIES LIMITED (GB) 1985-09-17 US disclosed
US-4486591-A CNS DISORDERS LILLY INDUSTRIES LIMITED (GB) 1984-12-04 US disclosed
US-4404137-A NEUROLEPTIC AGENTS; SEDATIVES; TRANQUILIZERS; ANTIEMETICS LILLY INDUSTRIES LIMITED (GB) 1983-09-13 US disclosed
EP-0027390-A1 Novel benzodiazepine compounds, their preparation, intermediates employed in their preparation, and pharmaceutical compositions containing them Lilly Industries Limited (GB) 1981-04-22 EP disclosed