SCHEMBL7273323

SCHEMBL7273323

N#CC1Cc2ccc(O)cc2C1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 8/20 0.46
DRD3 P35462 8/20 0.46
OPRK1 P41145 1/20 0.46
CYP11B2 P19099 2/20 0.44
CYP19A1 P11511 2/20 0.44
DRD4 P21917 6/20 0.42
CA1 P00915 2/20 0.39
CA2 P00918 2/20 0.39
ACHE P22303 2/20 0.39
HTR1A P08908 1/20 0.37
MEN1 O00255 1/20 0.37
ADRB2 P07550 1/20 0.37
CYP2D6 P10635 1/20 0.37
CASP1 P29466 1/20 0.37
KMT2A Q03164 1/20 0.37
CYP1A2 P05177 1/20 0.37
CYP11B1 P15538 1/20 0.37
PSEN1 P49768 1/20 0.37
PSEN2 P49810 1/20 0.37
APH1B Q8WW43 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9336168 0.76 MAPT (0.37) CYP11B2CA1CA2MEN1CASP1
SCHEMBL29833729 0.74 DRD2 (0.52) DRD2DRD3OPRK1CYP11B2CYP19A1
SCHEMBL11824507 0.74 DRD2 (0.52) DRD2DRD3OPRK1CYP11B2CYP19A1
SCHEMBL29539739 0.73 IDO1 (0.41) DRD3CYP11B2CYP1A2CYP11B1
SCHEMBL1415621 0.73 IDO1 (0.41) DRD3CYP11B2CYP1A2CYP11B1
SCHEMBL7274446 0.73 MAPT (0.51) CA1CA2
SCHEMBL13799411 0.72 DRD2 (0.50) DRD2DRD3OPRK1CYP11B2CYP19A1
SCHEMBL18350079 0.72 DRD2 (0.50) DRD2DRD3OPRK1CYP11B2CYP19A1
SCHEMBL25730011 0.72 DRD2 (0.50) DRD2DRD3OPRK1CYP11B2CYP19A1
SCHEMBL387649 0.72 DRD2 (0.71) DRD2DRD3OPRK1CYP11B2CYP19A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0483667-B1 Cyclic imino derivatives, process for their preparation and drugs containing them THOMAE GMBH DR K (DE) 1998-02-04 EP disclosed
US-5591769-A PYRROLIDINE DERIVATIVES; ANTICOAGULANTS KARL THOMAE GMBH (DE) 1997-01-07 US disclosed
US-5541343-A ANTIAGGLOMERANTS FOR CELLS OR ANTICOAGULANTS KARL THOMAE GMBH (DE) 1996-07-30 US disclosed
EP-0483667-A2 Cyclic imino derivatives, process for their preparation and drugs containing them Dr. Karl Thomae GmbH (DE) 1992-05-06 EP disclosed