SCHEMBL7273532

SCHEMBL7273532

O=CN(OCc1ccccc1)C(Cc1ccccc1)C(O)CCl

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABCB1 P08183 1/20 0.40
ALDH1A1 P00352 1/20 0.35
EPHX1 P07099 1/20 0.34
PPARG P37231 2/20 0.33
PPARA Q07869 2/20 0.33
CTSB P07858 2/20 0.33
CYP1A2 P05177 2/20 0.33
SLC1A3 P43003 2/20 0.33
SLC1A2 P43004 2/20 0.33
SLC1A1 P43005 2/20 0.33
TRPA1 O75762 1/20 0.33
MEN1 O00255 1/20 0.33
CYP2D6 P10635 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
KMT2A Q03164 1/20 0.33
CTRB1 P17538 2/20 0.33
SLC15A1 P46059 1/20 0.33
LTA4H P09960 1/20 0.33
LAP3 P28838 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7269426 0.93 PPARG (0.38) ABCB1ALDH1A1PPARGPPARAMEN1
SCHEMBL7267943 0.91 PPARG (0.41) ABCB1ALDH1A1PPARGPPARAKMT2A
SCHEMBL7289391 0.81 ABCB1 (0.39) ABCB1CTSBCYP1A2SLC1A3SLC1A2
SCHEMBL6925970 0.78 SLC15A1 (0.42) ABCB1EPHX1CYP1A2SLC1A3SLC1A2
SCHEMBL8660600 0.76 ABCB1 (0.37) ABCB1ALDH1A1CTSBMEN1KMT2A
SCHEMBL10686536 0.75 CYP1A2 (0.43) PPARGPPARACYP1A2SLC1A3SLC1A2
SCHEMBL10873777 0.73 SLC1A1 (0.45) ALDH1A1PPARGPPARACYP1A2SLC1A3
SCHEMBL10925477 0.72 EPHX1 (0.37) EPHX1CYP1A2SLC1A3SLC1A2SLC1A1
SCHEMBL7281228 0.72 AKT1 (0.43) ABCB1CTSB
SCHEMBL5275334 0.72 CSNK1E (0.49)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5652369-A PROTEASE INHIBITOR HOFFMANN-LA ROCHE INC. (US) 1997-07-29 US disclosed
US-5620987-A Amino acid derivatives HOFFMANN-LA ROCHE INC. (US) 1997-04-15 US disclosed
US-5554756-A PROTEASE INHIBITOR HOFFMANN-LA ROCHE INC. (US) 1996-09-10 US disclosed
US-5446161-A Protease inhibitor, viricides HOFFMANN-LA ROCHE INC. (US) 1995-08-29 US disclosed
EP-0346847-B1 Amino acid derivatives HOFFMANN LA ROCHE (CH) 1994-05-11 EP disclosed
US-5157041-A Viricides HOFFMANN-LA ROCHE INC. (US) 1992-10-20 US disclosed
EP-0346847-A2 Amino acid derivatives F. HOFFMANN-LA ROCHE AG (CH) 1989-12-20 EP disclosed