SCHEMBL7273947

SCHEMBL7273947

COC(=O)C[C@@H]1C[C@@H](COc2ccc(-c3ccc(C#N)cc3)cc2NC(C)=O)N(CCCc2ccccc2)C1=O

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EP300 Q09472 3/20 0.37
CHRNB2 P17787 1/20 0.35
CHRNB4 P30926 1/20 0.35
CHRNA3 P32297 1/20 0.35
CHRNA4 P43681 1/20 0.35
ABCB1 P08183 1/20 0.35
HPGD P15428 1/20 0.35
ABCG2 Q9UNQ0 1/20 0.35
ACLY P53396 1/20 0.34
HTR1A P08908 1/20 0.34
DRD4 P21917 1/20 0.34
HTR2A P28223 1/20 0.34
HRH1 P35367 1/20 0.34
OPRM1 P35372 1/20 0.34
LMNA P02545 2/20 0.34
MAPT P10636 2/20 0.34
ALDH1A1 P00352 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.33
MGAT2 Q10469 1/20 0.33
AR P10275 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7284181 0.91 ACLY (0.39) EP300ABCB1HPGDABCG2ACLY
SCHEMBL7280940 0.89 ABCB1 (0.36) EP300ABCB1HPGDABCG2HTR1A
SCHEMBL7274966 0.89 HRH3 (0.40) EP300ABCB1HPGDABCG2HTR1A
SCHEMBL7282659 0.89 ABCB1 (0.36) EP300ABCB1HPGDABCG2HTR1A
SCHEMBL7274992 0.88 ABCB1 (0.35) EP300ABCB1HPGDABCG2HTR1A
Hydrochloric Acid SCHEMBL7282362 0.88 PDE4A (0.37) CHRNB2CHRNB4CHRNA3CHRNA4LMNA
SCHEMBL7283703 0.87 ABCB1 (0.35) EP300ABCB1HPGDABCG2ACLY
SCHEMBL7273419 0.87 AR (0.39) EP300CHRNB2CHRNB4CHRNA3CHRNA4
SCHEMBL7281268 0.87 ABCB1 (0.44) ABCB1HPGDABCG2HTR1ADRD4
SCHEMBL7282551 0.87 ABCB1 (0.44) ABCB1HPGDABCG2HTR1ADRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0483667-B1 Cyclic imino derivatives, process for their preparation and drugs containing them THOMAE GMBH DR K (DE) 1998-02-04 EP disclosed
US-5591769-A PYRROLIDINE DERIVATIVES; ANTICOAGULANTS KARL THOMAE GMBH (DE) 1997-01-07 US disclosed
US-5541343-A ANTIAGGLOMERANTS FOR CELLS OR ANTICOAGULANTS KARL THOMAE GMBH (DE) 1996-07-30 US disclosed
EP-0483667-A2 Cyclic imino derivatives, process for their preparation and drugs containing them Dr. Karl Thomae GmbH (DE) 1992-05-06 EP disclosed