SCHEMBL7274258

SCHEMBL7274258

CC(C)(C)NC(=O)C1CN(C(=O)OC(C)(C)C)CCN1C(=O)OCc1ccccc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 2/20 0.54
TSHR P16473 2/20 0.54
KDM4E B2RXH2 2/20 0.54
LMNA P02545 2/20 0.54
TP53 P04637 1/20 0.54
GLA P06280 1/20 0.54
CYP3A4 P08684 1/20 0.54
CYP2D6 P10635 1/20 0.54
ADRA1D P25100 1/20 0.54
ADRA1A P35348 1/20 0.54
ADRA1B P35368 1/20 0.54
THPO P40225 1/20 0.54
HIF1A Q16665 1/20 0.54
HSD17B10 Q99714 1/20 0.54
GMNN O75496 1/20 0.54
ALDH1A1 P00352 1/20 0.54
MAPT P10636 1/20 0.54
HPGD P15428 1/20 0.54
MTOR P42345 1/20 0.54
PMP22 Q01453 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8865524 1.00 NPSR1 (0.54) NPSR1TSHRKDM4ELMNATP53
SCHEMBL9247790 0.96 PARP1 (0.54) NPSR1TSHRKDM4ELMNATP53
SCHEMBL375852 0.88 PDK1 (0.55) PDK1PDK2PDK3PDK4PARP1
SCHEMBL933923 0.88 PDK1 (0.55) PDK1PDK2PDK3PDK4PARP1
SCHEMBL2442588 0.88 PDK1 (0.55) PDK1PDK2PDK3PDK4PARP1
SCHEMBL5889141 0.88 CTRB1 (0.51) NPSR1TSHRKDM4ELMNAMAPT
SCHEMBL6487540 0.87 PDK1 (0.53) NPSR1MAPTPDK1PDK2PDK3
SCHEMBL1288345 0.87 PDK1 (0.53) NPSR1MAPTPDK1PDK2PDK3
SCHEMBL15298945 0.87 PDK1 (0.53) NPSR1MAPTPDK1PDK2PDK3
SCHEMBL7492256 0.87 PDK1 (0.54) PDK1PDK2PDK3PDK4PARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5652369-A PROTEASE INHIBITOR HOFFMANN-LA ROCHE INC. (US) 1997-07-29 US disclosed
US-5620987-A Amino acid derivatives HOFFMANN-LA ROCHE INC. (US) 1997-04-15 US disclosed
US-5554756-A PROTEASE INHIBITOR HOFFMANN-LA ROCHE INC. (US) 1996-09-10 US disclosed
US-5446161-A Protease inhibitor, viricides HOFFMANN-LA ROCHE INC. (US) 1995-08-29 US disclosed
EP-0346847-B1 Amino acid derivatives HOFFMANN LA ROCHE (CH) 1994-05-11 EP disclosed
US-5157041-A Viricides HOFFMANN-LA ROCHE INC. (US) 1992-10-20 US disclosed
EP-0346847-A2 Amino acid derivatives F. HOFFMANN-LA ROCHE AG (CH) 1989-12-20 EP disclosed