SCHEMBL7274340

SCHEMBL7274340

COc1ccc(CN2CC(OC(=O)O)CC2=O)cc1

nearest known ligand 0.60

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.54
CYP3A4 P08684 2/20 0.54
CYP2C19 P33261 2/20 0.54
L3MBTL1 Q9Y468 1/20 0.54
KMT2A Q03164 1/20 0.53
SMN1; SMN2 Q16637 3/20 0.50
MAPK1 P28482 2/20 0.49
ALOX15 P16050 1/20 0.49
MMP1 P03956 1/20 0.49
MMP13 P45452 1/20 0.49
LMNA P02545 1/20 0.48
CYP2D6 P10635 1/20 0.48
CYP2C9 P11712 1/20 0.48
HSD17B10 Q99714 1/20 0.47
GRM2 Q14416 1/20 0.46
HTT P42858 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28006519 0.90 ALDH1A1 (0.54) ALDH1A1CYP3A4CYP2C19L3MBTL1KMT2A
SCHEMBL7273770 0.89 CYP3A4 (0.55) ALDH1A1CYP3A4CYP2C19L3MBTL1KMT2A
SCHEMBL6612459 0.85 HTT (0.49) KMT2ASMN1; SMN2HTT
SCHEMBL6611174 0.85 HPGD (0.56) ALDH1A1KMT2ASMN1; SMN2LMNAHTT
SCHEMBL6609349 0.82 BTK (0.48) ALDH1A1KMT2ASMN1; SMN2MAPK1
SCHEMBL4095420 0.82 SMN1; SMN2 (0.73) ALDH1A1CYP3A4CYP2C19L3MBTL1KMT2A
SCHEMBL1710890 0.79 ALDH1A1 (0.65) ALDH1A1CYP3A4CYP2C19L3MBTL1KMT2A
SCHEMBL8348748 0.78 GRM2 (0.56) ALDH1A1CYP3A4CYP2C19L3MBTL1KMT2A
SCHEMBL1269684 0.78 CYP3A4 (0.67) ALDH1A1CYP3A4CYP2C19L3MBTL1KMT2A
SCHEMBL15415933 0.78 ALDH1A1 (0.64) ALDH1A1CYP3A4CYP2C19L3MBTL1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0483667-B1 Cyclic imino derivatives, process for their preparation and drugs containing them THOMAE GMBH DR K (DE) 1998-02-04 EP disclosed
EP-0483667-A2 Cyclic imino derivatives, process for their preparation and drugs containing them Dr. Karl Thomae GmbH (DE) 1992-05-06 EP disclosed