SCHEMBL7274353

SCHEMBL7274353

Cc1c(N)ccc2c1NC(=O)CC2(C)C

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.38
ALDH1A1 P00352 2/20 0.38
HPGD P15428 2/20 0.38
CYP19A1 P11511 2/20 0.37
RARB P10826 1/20 0.36
RARG P13631 1/20 0.36
BACE1 P56817 2/20 0.34
GLA P06280 2/20 0.33
GAA P10253 2/20 0.33
HSD17B10 Q99714 1/20 0.33
TYMS P04818 1/20 0.32
TSHR P16473 3/20 0.32
NPSR1 Q6W5P4 1/20 0.32
MEN1 O00255 1/20 0.31
MAPT P10636 1/20 0.31
ALOX15 P16050 1/20 0.31
CASP1 P29466 1/20 0.31
CASP7 P55210 1/20 0.31
KMT2A Q03164 1/20 0.31
HDAC3 O15379 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9379056 0.86 CYP19A1 (0.39) KDM4EALDH1A1HPGDCYP19A1RARB
SCHEMBL10587563 0.79 TYMS (0.38) CYP19A1RARBRARGBACE1TYMS
SCHEMBL6244091 0.79 ALDH1A1 (0.38) KDM4EALDH1A1HPGDRARBRARG
SCHEMBL7268304 0.78 BACE1 (0.33) CYP19A1RARBRARGBACE1
SCHEMBL5764522 0.74 PDE7A (0.46) KDM4EALDH1A1HPGDRARBRARG
SCHEMBL9379702 0.72 MAPK1 (0.38) ALDH1A1CYP19A1RARBRARGGAA
SCHEMBL7297952 0.71 CYP19A1 (0.36) KDM4EALDH1A1HPGDCYP19A1RARB
SCHEMBL3140413 0.69 CA9 (0.53) KDM4ECYP19A1RARBRARGBACE1
SCHEMBL17478594 0.69 PDE7A (0.45) ALDH1A1RARBRARGMEN1MAPT
SCHEMBL6432532 0.69 NR3C2 (0.56) KDM4EALDH1A1HPGDNPSR1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0322746-B1 Heterocyclic compounds ORION YHTYMAE OY (FI) 1996-05-29 EP disclosed
US-4963677-A TREATMENT OF CONGESTIVE HEART FAILURE ORION CORPORATION LTD. (FI) 1990-10-16 US disclosed
EP-0322746-A1 Heterocyclic compounds ORION CORPORATION LIMITED (FI) 1989-07-05 EP disclosed