SCHEMBL7274355

SCHEMBL7274355

Nc1cc(N)c(S)c(N)c1

nearest known ligand 0.38

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PTK2 Q05397 1/20 0.38
ALDH1A1 P00352 2/20 0.37
TSHR P16473 1/20 0.37
CYP3A4 P08684 3/20 0.35
TP53 P04637 1/20 0.35
CASP1 P29466 2/20 0.35
GAA P10253 2/20 0.33
MAPT P10636 1/20 0.33
KDM4E B2RXH2 1/20 0.32
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
THRB P10828 1/20 0.30
RECQL P46063 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24417902 0.84 ALDH1A1 (0.32) PTK2ALDH1A1TSHRCYP3A4TP53
SCHEMBL28770844 0.79 PTK2 (0.38) PTK2GAA
Hydrochloric Acid SCHEMBL28981675 0.76 PTK2 (0.35) PTK2
SCHEMBL21159438 0.73 ALDH1A1 (0.47) PTK2ALDH1A1TSHRCYP3A4TP53
SCHEMBL24418015 0.72 KDM4E (0.59) ALDH1A1CYP3A4CASP1GAAMAPT
SCHEMBL62068 0.67 KDM4E (0.45) ALDH1A1TSHRCYP3A4CASP1KDM4E
SCHEMBL2927013 0.67 CYP3A4 (0.58) ALDH1A1TSHRCYP3A4TP53CASP1
SCHEMBL24418016 0.67 PTK2 (0.41) PTK2ALDH1A1TSHRCYP3A4TP53
SCHEMBL9403002 0.67 PTK2 (0.40) PTK2ALDH1A1TSHRCYP3A4TP53
SCHEMBL62349 0.67

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0470514-B1 Carbostyril derivatives and pharmaceutical composition containing the same OTSUKA PHARMA CO LTD (JP) 1997-02-19 EP disclosed
US-5300513-A Vasopressin antagonists; vasodilators, hypotensive agents, water diuretics, and platelet agglutination inhibitors OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1994-04-05 US disclosed
EP-0470514-A1 Carbostyril derivatives and pharmaceutical composition containing the same OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1992-02-12 EP disclosed