SCHEMBL7274516

SCHEMBL7274516

CC(=O)Nc1c2c(nc3ccccc13)CCC(CCC1CCN(Cc3ccccc3)CC1)C2=O

nearest known ligand 0.53

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ACHE P22303 9/20 0.46
BCHE P06276 2/20 0.45
ALDH1A1 P00352 1/20 0.43
LMNA P02545 1/20 0.43
MAPT P10636 1/20 0.43
HTT P42858 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7281797 0.89 ACHE (0.46) ACHEBCHE
SCHEMBL7280234 0.88 ACHE (0.45) ACHEBCHEALDH1A1
SCHEMBL7282046 0.87 ACHE (0.46) ACHEBCHEHTT
SCHEMBL4501081 0.83 MEN1 (0.52) ACHE
Hydrochloric Acid SCHEMBL7279552 0.82 MEN1 (0.51) ACHE
SCHEMBL7273792 0.81 ACHE (0.42) ACHEALDH1A1
SCHEMBL7281819 0.81 ACHE (0.47) ACHEBCHE
SCHEMBL7272622 0.81 ACHE (0.52) ACHEBCHE
SCHEMBL7274046 0.80 ACHE (0.41) ACHEBCHEALDH1A1LMNAMAPT
Hydrochloric Acid SCHEMBL7279882 0.78 MEN1 (0.50) ACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0481429-B1 Quinoline derivatives SS PHARMACEUTICAL CO (JP) 2001-01-24 EP disclosed
EP-0987262-A1 Quinoline derivatives SS PHARMACEUTICAL CO., LTD. (JP) 2000-03-22 EP disclosed
US-5300517-A Treating Alzheimer's SS PHARMACEUTICAL CO., LTD. (JP) 1994-04-05 US disclosed
US-5240934-A Cognition activators SS PHARMACEUTICAL CO., LTD. (JP) 1993-08-31 US disclosed
US-5190951-A Inhibitors of acetylcholinesterase, treatment of senile dementia SS PHARMACEUTICAL CO., LTD. (JP) 1993-03-02 US disclosed
EP-0481429-A2 Quinoline derivatives SS PHARMACEUTICAL CO., LTD. (JP) 1992-04-22 EP disclosed