SCHEMBL7274557

SCHEMBL7274557

C=CC[C@@H]1C[C@@H](COc2cccc(CCCNC(=O)OC(C)(C)C)c2)N(CCCc2ccccc2)C1=O

nearest known ligand 0.44

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 3/20 0.44
MTNR1A P48039 2/20 0.37
MTNR1B P49286 2/20 0.37
ACACB O00763 1/20 0.37
FDFT1 P37268 2/20 0.37
CHRNB4 P30926 1/20 0.35
CHRNA3 P32297 1/20 0.35
CACNA1G O43497 1/20 0.35
MAPT P10636 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7281590 0.98 SIGMAR1 (0.44) SIGMAR1ACACBCACNA1G
SCHEMBL7283982 0.97 SIGMAR1 (0.43) SIGMAR1ACACBCHRNB4CHRNA3
SCHEMBL7284474 0.94 SIGMAR1 (0.41) SIGMAR1CHRNB4CHRNA3CACNA1G
SCHEMBL7283476 0.90 SIGMAR1 (0.45) SIGMAR1CACNA1G
SCHEMBL7280624 0.90 SIGMAR1 (0.45) SIGMAR1CHRNB4CHRNA3MAPT
SCHEMBL7274358 0.89 SIGMAR1 (0.44) SIGMAR1CACNA1G
SCHEMBL7282506 0.89 SIGMAR1 (0.45) SIGMAR1CACNA1G
SCHEMBL7275517 0.88 SIGMAR1 (0.43) SIGMAR1ACACB
SCHEMBL7282368 0.88 SIGMAR1 (0.44) SIGMAR1
SCHEMBL7283872 0.88 SIGMAR1 (0.44) SIGMAR1CACNA1G

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0483667-B1 Cyclic imino derivatives, process for their preparation and drugs containing them THOMAE GMBH DR K (DE) 1998-02-04 EP disclosed
US-5591769-A PYRROLIDINE DERIVATIVES; ANTICOAGULANTS KARL THOMAE GMBH (DE) 1997-01-07 US disclosed
US-5541343-A ANTIAGGLOMERANTS FOR CELLS OR ANTICOAGULANTS KARL THOMAE GMBH (DE) 1996-07-30 US disclosed
EP-0483667-A2 Cyclic imino derivatives, process for their preparation and drugs containing them Dr. Karl Thomae GmbH (DE) 1992-05-06 EP disclosed