SCHEMBL7275035

SCHEMBL7275035

Cc1ccc(S(=O)(=O)CC2CCC(=O)N2Cc2ccccc2)cc1

nearest known ligand 0.46

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.45
MEN1 O00255 1/20 0.45
CRBN Q96SW2 1/20 0.43
SMN1; SMN2 Q16637 3/20 0.42
LMNA P02545 2/20 0.42
NPC1 O15118 1/20 0.42
NR2F2 P24468 1/20 0.42
HTT P42858 1/20 0.42
RAB9A P51151 1/20 0.42
MCHR1 Q99705 1/20 0.42
GAA P10253 2/20 0.42
ALDH1A1 P00352 5/20 0.41
ELANE P08246 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41
TSHR P16473 1/20 0.40
KDM4E B2RXH2 1/20 0.40
MAPT P10636 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7275020 1.00 KMT2A (0.45) KMT2AMEN1CRBNSMN1; SMN2LMNA
SCHEMBL8534565 0.84 KMT2A (0.45) KMT2AMEN1SMN1; SMN2LMNAGAA
SCHEMBL8534561 0.82 KMT2A (0.43) KMT2AMEN1SMN1; SMN2LMNAGAA
SCHEMBL4374441 0.78 CRBN (0.50) CRBNSMN1; SMN2LMNANPC1NR2F2
SCHEMBL9621854 0.74 HCRTR2 (0.45) ALDH1A1CYP2C9CYP2C19TSHR
SCHEMBL6703838 0.74 TP53 (0.46) ALDH1A1CYP3A4CYP2C19TSHR
SCHEMBL27091866 0.74 KMT2A (0.58) KMT2AMEN1LMNAGAAALDH1A1
SCHEMBL16509689 0.73 MTNR1A (0.47) KMT2AMEN1ALDH1A1
SCHEMBL30829326 0.73 HCRTR1 (0.47) CYP3A4CYP2C19TSHR
SCHEMBL7275111 0.73 HCRTR1 (0.47) CYP3A4CYP2C19TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0381959-B1 Cyclohexaneacetamide derivatives HOFFMANN LA ROCHE (CH) 1995-05-03 EP disclosed
US-5015653-A Posess Cognitive Enhancement And Antiamnestic Activity HOFFMANN-LA ROCHE INC. (US) 1991-05-14 US disclosed
EP-0381959-A1 Cyclohexaneacetamide derivatives F. HOFFMANN-LA ROCHE AG (CH) 1990-08-16 EP disclosed