SCHEMBL7275066

SCHEMBL7275066

N=C(N)c1cnc(-c2ccc(OC[C@@H]3C[C@@H](CC(=O)O)C(=O)N3CC(=O)N3CCOCC3)cc2)nc1

nearest known ligand 0.43

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 2/20 0.43
ITGA2B P08514 2/20 0.43
USP2 O75604 2/20 0.38
ALDH1A1 P00352 5/20 0.37
NPC1 O15118 4/20 0.37
RAB9A P51151 3/20 0.37
HPGD P15428 3/20 0.37
TP53 P04637 2/20 0.37
KDM4E B2RXH2 2/20 0.37
SMN1; SMN2 Q16637 2/20 0.37
HSD17B10 Q99714 1/20 0.37
FKBP1A P62942 4/20 0.36
PTGS2 P35354 1/20 0.35
GRIN2B Q13224 3/20 0.35
LMNA P02545 2/20 0.35
GRIN1 Q05586 1/20 0.35
HTT P42858 1/20 0.35
ACHE P22303 1/20 0.34
POLB P06746 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7285404 0.92 ITGB3 (0.52) ITGB3ITGA2BUSP2ALDH1A1NPC1
Hydrochloric Acid SCHEMBL7284994 0.91 USP2 (0.39) ITGB3ITGA2BUSP2ALDH1A1NPC1
SCHEMBL7277654 0.91 ITGB3 (0.43) ITGB3ITGA2BALDH1A1LMNA
SCHEMBL7286629 0.90 ITGB3 (0.43) ITGB3ITGA2BALDH1A1LMNA
SCHEMBL7286641 0.90 ITGB3 (0.43) ITGB3ITGA2BALDH1A1LMNA
SCHEMBL7277653 0.89 ITGB3 (0.42) ITGB3ITGA2BLMNA
SCHEMBL7277402 0.88 ITGB3 (0.50) ITGB3ITGA2B
SCHEMBL7281127 0.84 ITGB3 (0.55) ITGB3ITGA2BALDH1A1LMNA
SCHEMBL7277794 0.84 ITGB3 (0.46) ITGB3ITGA2B
SCHEMBL7273817 0.83 ITGB3 (0.54) ITGB3ITGA2BALDH1A1LMNAACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5455348-A Anticoagulants Thomae, Karl (DE) 1995-10-03 US disclosed
EP-0528369-A2 Cyclic imino derivatives, pharmaceutical compositions containing them and process for their preparation Dr. Karl Thomae GmbH (DE) 1993-02-24 EP disclosed