SCHEMBL7276014

SCHEMBL7276014

COc1cc2cc(/C=N\O)sc2cc1OC

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
STING1 Q86WV6 14/20 0.42
ACHE P22303 2/20 0.40
TUBB4A P04350 2/20 0.39
TUBB P07437 2/20 0.39
TUBA3C P0DPH7 2/20 0.39
TUBA1B P68363 2/20 0.39
TUBA4A P68366 2/20 0.39
TUBB4B P68371 2/20 0.39
TUBB3 Q13509 2/20 0.39
TUBB2A Q13885 2/20 0.39
TUBB8 Q3ZCM7 2/20 0.39
TUBA3E Q6PEY2 2/20 0.39
TUBA1A Q71U36 2/20 0.39
TUBA1C Q9BQE3 2/20 0.39
TUBB6 Q9BUF5 2/20 0.39
TUBB2B Q9BVA1 2/20 0.39
TUBB1 Q9H4B7 2/20 0.39
HDAC3 O15379 1/20 0.37
HDAC4 P56524 1/20 0.37
HDAC1 Q13547 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7267085 1.00 STING1 (0.42) STING1ACHETUBB4ATUBBTUBA3C
SCHEMBL7267092 1.00 STING1 (0.42) STING1ACHETUBB4ATUBBTUBA3C
SCHEMBL9540978 0.83 MAPK1 (0.43) STING1HPGD
SCHEMBL9540983 0.83 MAPK1 (0.43) STING1HPGD
SCHEMBL9808648 0.78 CA2 (0.47) KDM4EHPGD
SCHEMBL7274175 0.78 BACE1 (0.53) TUBB4ATUBBTUBA3CTUBA1BTUBA4A
SCHEMBL7274183 0.78 BACE1 (0.53) TUBB4ATUBBTUBA3CTUBA1BTUBA4A
SCHEMBL7275954 0.78 BACE1 (0.53) TUBB4ATUBBTUBA3CTUBA1BTUBA4A
SCHEMBL7032634 0.77 CYP2A6 (0.51) STING1ACHEHDAC3HDAC4HDAC1
SCHEMBL7267852 0.74 HSD17B10 (0.39) STING1TUBB4ATUBBTUBA3CTUBA1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0352832-B1 COMPOUNDS WITH BRONCHODILATOR ACTIVITY AKZO N.V. (NL) 1992-05-06 EP disclosed
US-5026724-A Benzothiophene derivatives AKZO N.V. (NL) 1991-06-25 US disclosed
EP-0352832-A1 Compounds with bronchodilator activity AKZO N.V. (NL) 1990-01-31 EP disclosed