SCHEMBL7277196

SCHEMBL7277196

CCCn1c(=O)[nH]c(=O)c2[nH]c(C(C3CC3)C3CC3)nc21

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 6/20 0.71
ADORA2B P29275 6/20 0.71
ADORA1 P30542 2/20 0.60
ADORA3 P0DMS8 1/20 0.48
HPGD P15428 1/20 0.48
PDE4A P27815 1/20 0.48
BLM P54132 1/20 0.48
PDE4B Q07343 1/20 0.48
PDE4C Q08493 1/20 0.48
PDE4D Q08499 1/20 0.48
PDE3A Q14432 1/20 0.48
HSD17B10 Q99714 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7274376 0.88 ADORA2A (0.68) ADORA2AADORA2BADORA1
SCHEMBL2294590 0.83 ADORA2A (1.00) ADORA2AADORA2BADORA1ADORA3
SCHEMBL5226057 0.82 ADORA2A (0.56) ADORA2AADORA2BADORA1ADORA3HPGD
SCHEMBL30082250 0.81 ADORA2A (0.86) ADORA2AADORA2B
SCHEMBL7269959 0.80 ADORA2A (0.80) ADORA2AADORA2B
SCHEMBL8127160 0.79 ADORA2A (0.67) ADORA2AADORA2B
SCHEMBL7269624 0.78 ADORA2A (0.88) ADORA2AADORA2BADORA1ADORA3
SCHEMBL5227560 0.77 ADORA1 (0.90) ADORA2AADORA2BADORA1ADORA3
SCHEMBL9645551 0.75 ADORA1 (0.95) ADORA2AADORA2BADORA1ADORA3
SCHEMBL8118476 0.75 ADORA1 (1.00) ADORA2AADORA2BADORA1ADORA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0386675-B1 Xanthine derivatives KYOWA HAKKO KOGYO KK (JP) 1996-06-05 EP disclosed
US-5068236-A Diuretics, renal protective agents and hypotensives KYOWA HAKKO KOGYO CO., LTD. (JP) 1991-11-26 US disclosed
EP-0386675-A2 Xanthine derivatives KYOWA HAKKO KOGYO CO., LTD. (JP) 1990-09-12 EP disclosed