SCHEMBL7277354

SCHEMBL7277354

NC(=O)OC(Cc1ccc2ccccc2c1)C(O)CCl

nearest known ligand 0.44

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 1/20 0.43
HTR2C P28335 1/20 0.43
HTR2B P41595 1/20 0.43
PPARG P37231 2/20 0.41
PPARA Q07869 2/20 0.41
PPARD Q03181 1/20 0.41
SLC1A3 P43003 1/20 0.40
SLC1A2 P43004 1/20 0.40
SLC1A1 P43005 1/20 0.40
FCER2 P06734 2/20 0.40
TACR1 P25103 3/20 0.40
MMP9 P14780 1/20 0.39
DPP4 P27487 1/20 0.39
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
MC5R P33032 2/20 0.38
MC1R Q01726 2/20 0.38
EPHX1 P07099 1/20 0.38
CYP1A2 P05177 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7277361 1.00 HTR2A (0.43) HTR2AHTR2CHTR2BPPARGPPARA
SCHEMBL7291154 0.86 HTR2A (0.41) HTR2AHTR2CHTR2BPPARGPPARA
SCHEMBL27522583 0.83 SRR (0.42) PPARGPPARASLC1A3SLC1A2SLC1A1
SCHEMBL27522582 0.83 SRR (0.42) PPARGPPARASLC1A3SLC1A2SLC1A1
SCHEMBL4263442 0.83 SRR (0.42) PPARGPPARASLC1A3SLC1A2SLC1A1
SCHEMBL7291159 0.83 HTR2A (0.44) HTR2AHTR2CHTR2BPPARGPPARA
SCHEMBL7276239 0.77 PPARG (0.45) HTR2AHTR2CHTR2BPPARGPPARA
SCHEMBL7276245 0.77 PPARG (0.45) HTR2AHTR2CHTR2BPPARGPPARA
SCHEMBL7291165 0.77 HTR2A (0.39) HTR2AHTR2CHTR2BPPARGPPARA
SCHEMBL8918692 0.72 TACR1 (0.46) HTR2AHTR2CHTR2BFCER2TACR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5620987-A Amino acid derivatives HOFFMANN-LA ROCHE INC. (US) 1997-04-15 US disclosed
US-5554756-A PROTEASE INHIBITOR HOFFMANN-LA ROCHE INC. (US) 1996-09-10 US disclosed
EP-0346847-B1 Amino acid derivatives HOFFMANN LA ROCHE (CH) 1994-05-11 EP disclosed
US-5157041-A Viricides HOFFMANN-LA ROCHE INC. (US) 1992-10-20 US disclosed
EP-0346847-A2 Amino acid derivatives F. HOFFMANN-LA ROCHE AG (CH) 1989-12-20 EP disclosed