SCHEMBL7277601

SCHEMBL7277601

O=C1c2ccccc2C(=O)N1CN1CCCCC1

nearest known ligand 0.68

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CA1 P00915 3/20 0.68
CA2 P00918 3/20 0.68
ALDH1A1 P00352 7/20 0.53
TP53 P04637 1/20 0.53
GAA P10253 1/20 0.53
HPGD P15428 1/20 0.53
KMT2A Q03164 1/20 0.53
HSD17B10 Q99714 1/20 0.53
ACHE P22303 1/20 0.50
ALDH3A1 P30838 4/20 0.47
BCHE P06276 1/20 0.47
TERT O14746 1/20 0.46
METAP1 P53582 1/20 0.45
CA12 O43570 1/20 0.45
TSHR P16473 1/20 0.44
MAPK1 P28482 1/20 0.44
HTT P42858 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29619555 1.00 CA1 (0.68) CA1CA2ALDH1A1TP53GAA
SCHEMBL29097638 0.83 ALDH1A1 (0.69) ALDH1A1TP53GAAHPGDKMT2A
SCHEMBL3243125 0.83 ALDH1A1 (0.69) ALDH1A1TP53GAAHPGDKMT2A
Hydrochloric Acid SCHEMBL27677246 0.81 ALDH1A1 (0.67) ALDH1A1TP53GAAHPGDKMT2A
SCHEMBL26489650 0.81 ALDH1A1 (0.69) CA1CA2ALDH1A1GAAHPGD
SCHEMBL4609657 0.81 CA1 (1.00) CA1CA2ALDH1A1TP53ALDH3A1
SCHEMBL29163908 0.81 ALDH1A1 (0.66) ALDH1A1TP53GAAHPGDKMT2A
SCHEMBL30690126 0.81 ALDH1A1 (0.66) ALDH1A1TP53GAAHPGDKMT2A
SCHEMBL2362765 0.80 HTR1A (0.68) ACHE
SCHEMBL12124720 0.80 HTR1A (0.68)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0359311-B1 Butynylamine derivatives NIPPON SHINYAKU CO LTD (JP) 1997-01-15 EP disclosed
US-5036098-A Urogenital disorders NIPPON SHINYAKU CO., LTD. (JP) 1991-07-30 US disclosed
US-4927835-A ANTIPYRETICS NIPPON SHINYAKU CO., LTD. (JP) 1990-05-22 US disclosed
EP-0359311-A2 Butynylamine derivatives NIPPON SHINYAKU COMPANY, LIMITED (JP) 1990-03-21 EP disclosed
EP-0331195-A2 Acylphenol derivatives NIPPON SHINYAKU COMPANY, LIMITED (JP) 1989-09-06 EP disclosed
EP-0089055-B1 DEAZAPURINE DERIVATIVES Takeda Chemical Industries, Ltd. (JP) 1987-06-03 EP disclosed
US-4595530-A Thiodeazapurine derivatives TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1986-06-17 US disclosed
US-4571423-A Substituted 5-aminomethyl-2-acylaminopyrrolo[2,3-d]pyrimidin-4-ones TAKEDA CHEMICAL INDUSTRIES LTD. (JP) 1986-02-18 US disclosed
EP-0119591-A1 Thiodeazapurine derivatives Takeda Chemical Industries, Ltd. (JP) 1984-09-26 EP disclosed
EP-0089055-A2 Deazapurine derivatives Takeda Chemical Industries, Ltd. (JP) 1983-09-21 EP disclosed