SCHEMBL7277718

SCHEMBL7277718

O=C(CCc1ccccc1)C(F)(F)Cc1ccccc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KEAP1 Q14145 1/20 0.53
CES1 P23141 5/20 0.53
FAAH O00519 3/20 0.53
ALDH1A1 P00352 2/20 0.50
FFAR1 O14842 1/20 0.50
HDAC2 Q92769 2/20 0.47
HDAC8 Q9BY41 2/20 0.47
HDAC6 Q9UBN7 2/20 0.47
TDP1 Q9NUW8 1/20 0.47
GAA P10253 2/20 0.46
POLB P06746 1/20 0.46
HDAC1 Q13547 2/20 0.46
SMN1; SMN2 Q16637 2/20 0.46
HDAC3 O15379 1/20 0.46
MAPK1 P28482 1/20 0.46
ADRA1A P35348 1/20 0.46
HDAC4 P56524 1/20 0.46
SLC6A3 Q01959 1/20 0.46
HDAC7 Q8WUI4 1/20 0.46
HDAC10 Q969S8 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7460240 0.85 KEAP1 (0.53) KEAP1CES1FAAHALDH1A1FFAR1
SCHEMBL1274684 0.82 CES1 (0.73) KEAP1CES1FAAHALDH1A1FFAR1
SCHEMBL5598343 0.81 KEAP1 (0.57) KEAP1CES1FAAHALDH1A1FFAR1
SCHEMBL11546063 0.81 CES1 (0.52) KEAP1CES1FAAHALDH1A1SMN1; SMN2
SCHEMBL9767789 0.80 CES1 (0.47) KEAP1CES1FAAHALDH1A1FFAR1
SCHEMBL7808017 0.79 KEAP1 (0.55) KEAP1CES1FAAHALDH1A1FFAR1
SCHEMBL17048769 0.79 CES1 (0.50) KEAP1CES1FAAHALDH1A1HDAC2
SCHEMBL28345545 0.79 KEAP1 (0.55) KEAP1CES1FAAHALDH1A1FFAR1
SCHEMBL5235928 0.78 SMN1; SMN2 (0.57) KEAP1CES1FAAHSMN1; SMN2HIF1A
SCHEMBL29187270 0.78 KEAP1 (0.53) KEAP1CES1FAAHALDH1A1FFAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0839798-A2 Intermediates for preparating non-peptide retroviral protease inhibitors ABBOTT LABORATORIES (US) 1998-05-06 EP disclosed
US-5670675-A Retroviral protease inhibiting compounds ABBOTT LABORATORIES (US) 1997-09-23 US disclosed
US-5545750-A TREATING HUMAN IMMUNODEFICIENCY VIRUS ABBOTT LABORATORIES (US) 1996-08-13 US disclosed
US-5142056-A Human immunodeficiency virus protease inhibitor ABBOTT LABORATORIES (US) 1992-08-25 US disclosed
EP-0402646-A1 Retroviral protease inhibiting compounds ABBOTT LABORATORIES (US) 1990-12-19 EP disclosed