SCHEMBL28345545

SCHEMBL28345545

O=C(CCc1ccccc1)C(F)(F)I

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KEAP1 Q14145 1/20 0.55
CES1 P23141 5/20 0.54
FAAH O00519 3/20 0.54
ALDH1A1 P00352 2/20 0.52
FFAR1 O14842 1/20 0.52
HDAC2 Q92769 2/20 0.48
HDAC8 Q9BY41 2/20 0.48
HDAC6 Q9UBN7 2/20 0.48
TDP1 Q9NUW8 1/20 0.48
POLB P06746 1/20 0.47
GAA P10253 1/20 0.47
GPR52 Q9Y2T5 1/20 0.47
HDAC1 Q13547 2/20 0.47
HDAC3 O15379 1/20 0.47
MAPK1 P28482 1/20 0.47
ADRA1A P35348 1/20 0.47
HDAC4 P56524 1/20 0.47
SLC6A3 Q01959 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
HDAC7 Q8WUI4 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1274684 0.84 CES1 (0.73) KEAP1CES1FAAHALDH1A1FFAR1
SCHEMBL7808017 0.81 KEAP1 (0.55) KEAP1CES1FAAHALDH1A1FFAR1
SCHEMBL7277718 0.79 KEAP1 (0.53) KEAP1CES1FAAHALDH1A1FFAR1
SCHEMBL7460240 0.79 KEAP1 (0.53) KEAP1CES1FAAHALDH1A1FFAR1
SCHEMBL9770696 0.78 KEAP1 (0.52) KEAP1CES1FAAHALDH1A1FFAR1
SCHEMBL28460352 0.76 KEAP1 (0.59) KEAP1CES1FAAHALDH1A1FFAR1
Phenyl Propionic Acid SCHEMBL27428011 0.76 KEAP1 (0.79) KEAP1CES1FAAHALDH1A1FFAR1
SCHEMBL5598351 0.76 ALDH1A1 (0.61) KEAP1CES1FAAHALDH1A1FFAR1
SCHEMBL8153818 0.76 ALDH1A1 (0.61) KEAP1CES1FAAHALDH1A1FFAR1
SCHEMBL15562490 0.76 ALDH1A1 (0.55) KEAP1CES1FAAHALDH1A1FFAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110683943-B Fluoro 1, 3-eneyne compound and preparation method thereof 上海应用技术大学 2023-03-31 CN disclosed
CN-113548936-A Aroyldifluoromethyl olefin and preparation method thereof 上海应用技术大学 2021-10-26 CN disclosed
CN-110683943-A Fluoro 1, 3-eneyne compound and preparation method thereof 上海应用技术大学 2020-01-14 CN disclosed