SCHEMBL7278752

SCHEMBL7278752

COC(=O)c1ccc(Cn2cnc3c4cccnc4n(-c4ccccc4)c(=O)c32)cc1

nearest known ligand 0.74

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 7/20 0.74
PDE4B Q07343 5/20 0.64
PDE4C Q08493 5/20 0.64
PDE4D Q08499 5/20 0.64
MAPK8 P45983 6/20 0.46
MMP13 P45452 1/20 0.46
YTHDC1 Q96MU7 1/20 0.46
RECQL P46063 1/20 0.45
MAPK10 P53779 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
POLB P06746 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7281463 0.87 PDE4A (0.80) PDE4APDE4BPDE4CPDE4DPOLB
SCHEMBL7272788 0.86 PDE4A (1.00) PDE4APDE4BPDE4CPDE4DSMN1; SMN2
SCHEMBL7279910 0.85 PDE4A (0.85) PDE4APDE4BPDE4CPDE4DSMN1; SMN2
SCHEMBL7281912 0.84 PDE4A (0.87) PDE4APDE4BPDE4CPDE4DSMN1; SMN2
SCHEMBL7271255 0.83 PDE4A (0.85) PDE4APDE4BPDE4CPDE4DSMN1; SMN2
SCHEMBL7272860 0.83 PDE4A (0.80) PDE4APDE4BPDE4CPDE4D
SCHEMBL7271311 0.81 PDE4A (0.85) PDE4APDE4BPDE4CPDE4DSMN1; SMN2
SCHEMBL7338034 0.81 PDE4A (0.77) PDE4APDE4BPDE4CPDE4DPOLB
SCHEMBL7278166 0.80 PDE4A (0.76) PDE4APDE4BPDE4CPDE4DPOLB
SCHEMBL7271125 0.80 PDE4A (0.79) PDE4APDE4BPDE4CPDE4D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0459505-B1 Imidazonaphthyridine derivatives KYOWA HAKKO KOGYO KK (JP) 1996-10-02 EP disclosed
US-5536730-A ANTIINFLAMMATORY, ANTIALLERGIC AND BRONCHODILATIVE ACTIVITY KYOWA HAKKO KOGYO CO. LTD. (JP) 1996-07-16 US disclosed
US-5468756-A Antiinflammatory, antiallergen KYOWA HAKKO KOGYO CO., LTD. (JP) 1995-11-21 US disclosed
US-5364859-A Antiinflammatory agents, antiallergens, bronchodilators KYOWA HAKKO KOGYO CO., LTD. (JP) 1994-11-15 US disclosed
EP-0459505-A1 Imidazonaphthyridine derivatives KYOWA HAKKO KOGYO CO., LTD. (JP) 1991-12-04 EP disclosed