SCHEMBL72789

SCHEMBL72789

CC(=O)Nc1cccc(-c2cnc3ccccn23)c1

nearest known ligand 0.63

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
FYN P06241 15/20 0.63
DYRK3 O43781 1/20 0.58
CCNT1 O60563 1/20 0.58
CCNA2 P20248 1/20 0.58
CDK2 P24941 1/20 0.58
CDK9 P50750 1/20 0.58
CDK5 Q00535 1/20 0.58
DYRK1A Q13627 1/20 0.58
CDK5R1 Q15078 1/20 0.58
DYRK2 Q92630 1/20 0.58
DYRK1B Q9Y463 1/20 0.58
KDM4E B2RXH2 1/20 0.57
ALDH1A1 P00352 1/20 0.57
SMN1; SMN2 Q16637 1/20 0.57
FGFR3 P22607 2/20 0.57
KDR P35968 2/20 0.57
RIPK2 O43353 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13336637 0.87 KDR (0.67) FYNFGFR3KDR
Hydrochloric Acid SCHEMBL3321535 0.86 KDR (0.66) FYNFGFR3KDR
SCHEMBL73833 0.85 FGFR3 (0.73) FGFR3KDR
SCHEMBL3325195 0.84 FGFR3 (0.79) FYNDYRK3CCNT1CCNA2CDK2
SCHEMBL3323066 0.84 FYN (0.65) FYNDYRK3CCNT1CCNA2CDK2
SCHEMBL23535614 0.82 FYN (0.65) FYNDYRK3CCNT1CCNA2CDK2
SCHEMBL30006622 0.82 FYN (0.65) FYNDYRK3CCNT1CCNA2CDK2
SCHEMBL13336397 0.82 FYN (0.64) FYNDYRK3CCNT1CCNA2CDK2
SCHEMBL3323050 0.82 KDR (0.69) FYNFGFR3KDR
SCHEMBL3323645 0.81 KDR (0.81) FGFR3KDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8131527-B1 FGFR pharmacophore compounds ASTEX THERAPEUTICS LTD. (GB) 2012-03-06 US disclosed
US-8131527-B1 FGFR pharmacophore compounds ASTEX THERAPEUTICS LTD. (GB) 2012-03-06 US disclosed