SCHEMBL7278992

SCHEMBL7278992

NC(=O)C(c1ccc(Cl)cc1)N1CCNCC1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 1/20 0.58
CYP19A1 P11511 1/20 0.58
OPRD1 P41143 4/20 0.49
OPRM1 P35372 1/20 0.49
NSD2 O96028 1/20 0.47
CHEK2 O96017 1/20 0.45
HTR3E A5X5Y0 1/20 0.42
HTR3B O95264 1/20 0.42
ADRB1 P08588 1/20 0.42
HTR3A P46098 1/20 0.42
HTR3D Q70Z44 1/20 0.42
HTR3C Q8WXA8 1/20 0.42
SIGMAR1 Q99720 1/20 0.42
ADRB2 P07550 2/20 0.42
NPSR1 Q6W5P4 1/20 0.42
MAPT P10636 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.40
SLC6A2 P23975 2/20 0.40
SLC6A4 P31645 2/20 0.40
ALDH1A1 P00352 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7278715 0.84 OPRD1 (0.50) CYP2D6CYP19A1OPRD1OPRM1ADRB1
SCHEMBL793646 0.84 OPRD1 (0.60) OPRD1OPRM1SLC6A2SLC6A4
SCHEMBL7282376 0.82 SLC6A4 (0.49) CYP2D6CYP19A1OPRD1HTR3EHTR3B
SCHEMBL15797474 0.81 SMN1; SMN2 (0.59) NSD2ADRB2SMN1; SMN2ALDH1A1
SCHEMBL25083517 0.81 CYP2D6 (0.54) CYP2D6CYP19A1OPRD1OPRM1CHEK2
SCHEMBL7282015 0.81 TEAD1 (0.53) OPRD1SLC6A4
SCHEMBL7288846 0.81 CHRM2 (0.55) CYP2D6OPRD1OPRM1HTR3EHTR3B
SCHEMBL7279116 0.81 OPRD1 (0.44) CYP2D6CYP19A1OPRD1OPRM1SLC6A4
Hydrochloric Acid SCHEMBL29894729 0.80 CYP2D6 (0.53) CYP2D6CYP19A1OPRD1OPRM1HTR3E
SCHEMBL7289405 0.80 CHRM2 (0.49) CYP2D6CYP19A1OPRD1OPRM1SLC6A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4567264-A ADRENERGIC BLOCKING AGENTS SYNTEX (U.S.A.) INC. (US) 1986-01-28 US disclosed
EP-0126449-A1 Cardioselective aryloxy- and arylthio-hydroxypropyl piperazinyl acetanilides wich affect calcium entry SYNTEX (U.S.A.) INC. (US) 1984-11-28 EP disclosed