SCHEMBL7279562

SCHEMBL7279562

CCCS(=O)(=O)c1ccc(-c2nc3cnccc3[nH]2)c(OC)c1

nearest known ligand 0.49

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 10/20 0.49
CYP3A4 P08684 9/20 0.49
PDE5A O76074 6/20 0.49
CYP2D6 P10635 4/20 0.49
PDE3B Q13370 1/20 0.49
PDE3A Q14432 1/20 0.49
CYP2C19 P33261 9/20 0.47
CYP1A2 P05177 8/20 0.47
KDM4E B2RXH2 1/20 0.39
ALDH1A1 P00352 1/20 0.39
HPGD P15428 1/20 0.39
AAK1 Q2M2I8 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7272031 0.86 PDE5A (0.54) PDE5APDE3BPDE3AKDM4EALDH1A1
SCHEMBL7272060 0.85 PDE5A (0.45) CYP2C9CYP3A4PDE5ACYP2D6PDE3B
Hydrochloric Acid SCHEMBL10859310 0.84 PDE5A (0.52) PDE5APDE3BPDE3ACYP1A2KDM4E
SCHEMBL7279838 0.83 CYP1A2 (0.43) CYP2C9CYP3A4PDE5ACYP2D6PDE3B
SCHEMBL11018071 0.81 CYP2C9 (0.47) CYP2C9CYP3A4PDE5ACYP2D6PDE3B
SCHEMBL9634654 0.79 PDE5A (0.53) PDE5APDE3BPDE3ACYP1A2KDM4E
SCHEMBL11018077 0.79 CYP2C9 (0.54) CYP2C9CYP3A4CYP2D6CYP2C19CYP1A2
SCHEMBL10748751 0.79 PDE5A (0.51) PDE5APDE3BPDE3ACYP1A2KDM4E
SCHEMBL11065268 0.78 CYP2C9 (0.44) CYP2C9CYP3A4PDE5ACYP2D6CYP2C19
SCHEMBL10744182 0.78 PDE5A (0.52) CYP3A4PDE5APDE3BPDE3ACYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4904785-A INOTROPIC AGENTS FOR CARDIOVASCULAR DISORDERS ELI LILLY AND COMPANY (US) 1990-02-27 US disclosed
US-4758574-A 2-phenylimidazio (4,5-c) pyridines ELI LILLY AND COMPANY (US) 1988-07-19 US disclosed
EP-0093593-A2 Pyridine compounds ELI LILLY AND COMPANY (US) 1983-11-09 EP disclosed