SCHEMBL11018071

SCHEMBL11018071

CCCS(=O)(=O)c1ccc(-c2nc3cc(C#N)ccc3[nH]2)c(OC)c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 7/20 0.47
CYP3A4 P08684 6/20 0.47
CYP2D6 P10635 2/20 0.47
CYP2C19 P33261 6/20 0.45
CYP1A2 P05177 5/20 0.45
MAPK10 P53779 1/20 0.40
CA12 O43570 1/20 0.40
CA1 P00915 1/20 0.40
CA2 P00918 1/20 0.40
CA9 Q16790 1/20 0.40
PTGDR2 Q9Y5Y4 2/20 0.40
PDE5A O76074 1/20 0.36
PDE3B Q13370 1/20 0.36
PDE3A Q14432 1/20 0.36
ALK Q9UM73 2/20 0.36
AMY1A P0DUB6 1/20 0.36
SCN9A Q15858 1/20 0.36
FLT1 P17948 1/20 0.35
FLT4 P35916 1/20 0.35
KDR P35968 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10763275 0.93 MAPK10 (0.42) CYP2C9CYP3A4CYP2D6CYP2C19CYP1A2
SCHEMBL11018077 0.92 CYP2C9 (0.54) CYP2C9CYP3A4CYP2D6CYP2C19CYP1A2
SCHEMBL11017633 0.88 ALDH1A1 (0.44) MAPK10CA12CA1CA2CA9
SCHEMBL11021893 0.87 ATR (0.44) MAPK10CA12CA1CA2CA9
SCHEMBL11020313 0.86 CA2 (0.54) MAPK10CA12CA1CA2CA9
SCHEMBL11021552 0.86 L3MBTL1 (0.47) MAPK10CA12CA1CA2CA9
SCHEMBL11018186 0.85 CYP3A4 (0.48) CYP2C9CYP3A4CYP2D6CYP2C19CYP1A2
SCHEMBL11016112 0.84 SCN9A (0.42) MAPK10CA12CA1CA2CA9
SCHEMBL11018857 0.84 MAPT (0.44) MAPK10CA12CA1CA2CA9
SCHEMBL7279562 0.81 CYP2C9 (0.49) CYP2C9CYP3A4CYP2D6CYP2C19CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0148431-A1 Benzimidazoles, their preparation, and medicaments containing these compounds Dr. Karl Thomae GmbH (DE) 1985-07-17 EP disclosed