SCHEMBL11018077

SCHEMBL11018077

CCCS(=O)(=O)c1ccc(-c2nc3ccc(C#N)cc3[nH]2)c(OC)c1

nearest known ligand 0.54

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 12/20 0.54
CYP3A4 P08684 11/20 0.54
CYP2D6 P10635 5/20 0.54
CYP2C19 P33261 11/20 0.53
CYP1A2 P05177 10/20 0.53
ATR Q13535 1/20 0.43
PKN1 Q16512 1/20 0.42
PKN2 Q16513 1/20 0.42
CFB P00751 3/20 0.41
CHEK2 O96017 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11018186 0.93 CYP3A4 (0.48) CYP2C9CYP3A4CYP2D6CYP2C19CYP1A2
SCHEMBL11018071 0.92 CYP2C9 (0.47) CYP2C9CYP3A4CYP2D6CYP2C19CYP1A2
SCHEMBL11017639 0.88 MAPT (0.49) CYP2C9CYP3A4CYP2D6ATRPKN1
SCHEMBL11021898 0.87 ATR (0.53) ATRPKN1PKN2CFBCHEK2
SCHEMBL11020318 0.86 CA12 (0.54) ATRPKN1PKN2CFBCHEK2
SCHEMBL11021561 0.86 L3MBTL1 (0.47) CYP2C9CYP3A4CYP2D6ATRPKN1
SCHEMBL10763275 0.85 MAPK10 (0.42) CYP2C9CYP3A4CYP2D6CYP2C19CYP1A2
SCHEMBL11018866 0.84 MAPT (0.44) ATRPKN1PKN2CFBCHEK2
SCHEMBL11016115 0.84 CFB (0.47) ATRPKN1PKN2CFBCHEK2
SCHEMBL11017633 0.80 ALDH1A1 (0.44)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0148431-A1 Benzimidazoles, their preparation, and medicaments containing these compounds Dr. Karl Thomae GmbH (DE) 1985-07-17 EP disclosed