SCHEMBL7279657

SCHEMBL7279657

Cc1cccc(-n2c(=O)c3[nH]cnc3c3cccnc32)c1

nearest known ligand 0.74

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 7/20 0.74
PDE4B Q07343 7/20 0.74
PDE4D Q08499 7/20 0.74
PDE4C Q08493 6/20 0.74
POLB P06746 1/20 0.42
PDE1A P54750 1/20 0.40
PDE1B Q01064 1/20 0.40
LMNA P02545 3/20 0.39
ALDH1A1 P00352 2/20 0.39
KMT2A Q03164 2/20 0.39
MAPT P10636 1/20 0.39
PPARG P37231 1/20 0.39
RXFP1 Q9HBX9 1/20 0.39
NR2E3 Q9Y5X4 1/20 0.39
NCOR2 Q9Y618 1/20 0.39
HPGD P15428 3/20 0.39
KDM4E B2RXH2 1/20 0.39
S1PR4 O95977 1/20 0.39
GLA P06280 1/20 0.39
GAA P10253 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7273701 0.87 PDE4A (0.76) PDE4APDE4BPDE4DPDE4CPDE1A
SCHEMBL7280371 0.87 PDE4A (0.79) PDE4APDE4BPDE4DPDE4CPOLB
SCHEMBL7328426 0.86 PDE4A (0.71) PDE4APDE4BPDE4DPDE4CPOLB
SCHEMBL7271411 0.85 PDE4A (1.00) PDE4APDE4BPDE4DPDE4CPDE1A
SCHEMBL7340105 0.79 PDE4A (0.74) PDE4APDE4BPDE4DPDE4CPDE1A
SCHEMBL2457079 0.75 PDE4A (0.81) PDE4APDE4BPDE4DPDE4CPDE1A
SCHEMBL7278448 0.73 PDE4A (0.52) PDE4APDE4BPDE4DPDE4CPOLB
SCHEMBL7270964 0.72 PDE4A (0.79) PDE4APDE4BPDE4DPDE4CPOLB
SCHEMBL7278555 0.72 POLB (0.43) PDE4APDE4BPDE4DPDE4CPOLB
SCHEMBL7271034 0.71 PDE4A (0.80) PDE4APDE4BPDE4DPDE4CPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0459505-B1 Imidazonaphthyridine derivatives KYOWA HAKKO KOGYO KK (JP) 1996-10-02 EP disclosed
US-5536730-A ANTIINFLAMMATORY, ANTIALLERGIC AND BRONCHODILATIVE ACTIVITY KYOWA HAKKO KOGYO CO. LTD. (JP) 1996-07-16 US disclosed
US-5468756-A Antiinflammatory, antiallergen KYOWA HAKKO KOGYO CO., LTD. (JP) 1995-11-21 US disclosed
US-5364859-A Antiinflammatory agents, antiallergens, bronchodilators KYOWA HAKKO KOGYO CO., LTD. (JP) 1994-11-15 US disclosed
EP-0459505-A1 Imidazonaphthyridine derivatives KYOWA HAKKO KOGYO CO., LTD. (JP) 1991-12-04 EP disclosed