SCHEMBL7273701

SCHEMBL7273701

O=c1c2[nH]cnc2c2cccnc2n1-c1cccc(Cl)c1

nearest known ligand 0.76

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 10/20 0.76
PDE4B Q07343 8/20 0.76
PDE4C Q08493 8/20 0.76
PDE4D Q08499 8/20 0.76
MAPT P10636 3/20 0.51
HPGD P15428 2/20 0.51
MEN1 O00255 1/20 0.51
CYP1A2 P05177 1/20 0.51
CYP2C19 P33261 1/20 0.51
KMT2A Q03164 1/20 0.51
KDM4E B2RXH2 1/20 0.41
GAA P10253 1/20 0.41
PDE1A P54750 1/20 0.41
PDE1B Q01064 1/20 0.41
RPS6KB1 P23443 1/20 0.39
FEN1 P39748 1/20 0.39
AURKA O14965 1/20 0.38
DAPK3 O43293 1/20 0.38
JAK2 O60674 1/20 0.38
PRKD3 O94806 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7279657 0.87 PDE4A (0.74) PDE4APDE4BPDE4CPDE4DMAPT
SCHEMBL7271411 0.86 PDE4A (1.00) PDE4APDE4BPDE4CPDE4DCYP2C19
SCHEMBL7328426 0.85 PDE4A (0.71) PDE4APDE4BPDE4CPDE4DMAPT
SCHEMBL7280371 0.81 PDE4A (0.79) PDE4APDE4BPDE4CPDE4DHPGD
SCHEMBL7340105 0.78 PDE4A (0.74) PDE4APDE4BPDE4CPDE4DMAPT
SCHEMBL2457079 0.76 PDE4A (0.81) PDE4APDE4BPDE4CPDE4DHPGD
SCHEMBL9267553 0.75 MAPT (0.47) PDE4APDE4BPDE4CPDE4DMAPT
SCHEMBL9132147 0.75 MAPT (0.52) PDE4APDE4BPDE4CPDE4DMAPT
SCHEMBL5249954 0.74 HPGD (0.64) PDE4BPDE4DMAPTHPGDMEN1
SCHEMBL10427752 0.73 KMT2A (0.50) PDE4APDE4BPDE4CPDE4DMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0459505-B1 Imidazonaphthyridine derivatives KYOWA HAKKO KOGYO KK (JP) 1996-10-02 EP disclosed
US-5536730-A ANTIINFLAMMATORY, ANTIALLERGIC AND BRONCHODILATIVE ACTIVITY KYOWA HAKKO KOGYO CO. LTD. (JP) 1996-07-16 US disclosed
US-5468756-A Antiinflammatory, antiallergen KYOWA HAKKO KOGYO CO., LTD. (JP) 1995-11-21 US disclosed
US-5364859-A Antiinflammatory agents, antiallergens, bronchodilators KYOWA HAKKO KOGYO CO., LTD. (JP) 1994-11-15 US disclosed
EP-0459505-A1 Imidazonaphthyridine derivatives KYOWA HAKKO KOGYO CO., LTD. (JP) 1991-12-04 EP disclosed