Perflenapent

Perflenapent

SCHEMBL727982

CC[N+](CC)(CC)CC.FC(F)(F)C(F)(F)C(F)(F)C(F)(F)C(F)(F)F

nearest known ligand 0.50

Full drug profile on Sugi Atlas →

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.50
NFKB1 P19838 1/20 0.50
KCNA1 Q09470 1/20 0.50
KDM4E B2RXH2 1/20 0.47
PMP22 Q01453 1/20 0.47
ATM Q13315 1/20 0.47
LMNA P02545 1/20 0.38
THRB P10828 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Tetrylammonium SCHEMBL1183170 1.00 TSHR (0.50) TSHRNFKB1KCNA1KDM4EPMP22
Perflexane SCHEMBL727759 1.00 TSHR (0.50) TSHRNFKB1KCNA1KDM4EPMP22
Tetrylammonium SCHEMBL727741 1.00 TSHR (0.50) TSHRNFKB1KCNA1KDM4EPMP22
Perflubutane SCHEMBL1490719 0.97 TSHR (0.53) TSHRNFKB1KCNA1KDM4EPMP22
Perflutren SCHEMBL729416 0.90 TSHR (0.53) TSHRNFKB1KCNA1KDM4EPMP22
Tetrylammonium SCHEMBL727439 0.83 TSHR (0.61) TSHRNFKB1KCNA1KDM4EPMP22
Tetrylammonium SCHEMBL20237361 0.80 TSHR (0.42) TSHRNFKB1KCNA1KDM4EPMP22
Tetrylammonium SCHEMBL727740 0.79 TSHR (0.67) TSHRNFKB1KCNA1KDM4EPMP22
Hydrogen Sulfide SCHEMBL28468639 0.75 LMNA (0.57) LMNATHRB
Hydrogen Sulfide SCHEMBL28956837 0.75 LMNA (0.57) LMNATHRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 35 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2294135-B1 FLAME RETARDANT, OPTICALLY CLEAR THERMOPLASTIC MOLDING COMPOSITION COVESTRO LLC (US) 2017-07-26 EP claimed
EP-2480608-B1 FLAME RETARDANT, OPTICALLY CLEAR THERMOPLASTIC MOLDING COMPOSITION COVESTRO LLC (US) 2017-05-24 EP claimed
EP-2480608-A2 FLAME RETARDANT, OPTICALLY CLEAR THERMOPLASTIC MOLDING COMPOSITION Bayer MaterialScience LLC (US) 2012-08-01 EP claimed
JP-2011526942-A 2011-10-20 JP claimed
WO-2011037611-A2 FLAME RETARDANT, OPTICALLY CLEAR THERMOPLASTIC MOLDING COMPOSITION BAYER MATERIALSCIENCE LLC (US) 2011-03-31 WO claimed
US-20110071241-A1 FLAME RETARDANT, OPTICALLY CLEAR THERMOPLASTIC MOLDING COMPOSITION BAYER MATERIALSCIENCE LLC (US) 2011-03-24 US claimed
EP-2294135-A2 FLAME RETARDANT, OPTICALLY CLEAR THERMOPLASTIC MOLDING COMPOSITION Bayer MaterialScience LLC (US) 2011-03-16 EP claimed
WO-2010005486-A2 FLAME RETARDANT, OPTICALLY CLEAR THERMOPLASTIC MOLDING COMPOSITION BAYER MATERIALSCIENCE LLC (US) 2010-01-14 WO claimed
US-20090326129-A1 Flame retardant, optically clear thermoplastic molding composition BAYER MATERIALSCIENCE LLC 2009-12-31 US claimed
US-7288579-B2 Method for reducing haze in a fire resistant polycarbonate composition GENERAL ELECTRIC COMPANY (US) 2007-10-30 US claimed
EP-1702005-B1 POLYCARBONATE COMPOSITION GEN ELECTRIC (US) 2007-07-25 EP claimed
US-20040132865-A1 Method for reducing haze in a fire resistant polycarbonate composition SABIC INNOVATIVE PLASTICS IP B.V. (NL) 2004-07-08 US claimed
JP-2004516376-A 2004-06-03 JP claimed
US-6730720-B2 BLENDING A FLAME RETARDANT SALT WITH A POLYCARBONATE TO PRODUCE A CONCENTRATE AND THEN BLENDING THE CONCENTRATE WITH A POLYCARBONATE TO FORM A TRANSPARENT POLYCARBONATE BLEND GENERAL ELECTRIC COMPANY 2004-05-04 US claimed
US-20020123544-A1 Method for reducing haze in a fire resistant polycarbonate composition SABIC INNOVATIVE PLASTICS IP B.V. (NL) 2002-09-05 US claimed
WO-2002051923-A2 METHOD FOR REDUCING HAZE IN A FIRE RESISTANT POLYCARBONATE COMPOSITION GENERAL ELECTRIC COMPANY (US) 2002-07-04 WO claimed
EP-2294135-B1 FLAME RETARDANT, OPTICALLY CLEAR THERMOPLASTIC MOLDING COMPOSITION COVESTRO LLC (US) 2017-07-26 EP disclosed
EP-2480608-B1 FLAME RETARDANT, OPTICALLY CLEAR THERMOPLASTIC MOLDING COMPOSITION COVESTRO LLC (US) 2017-05-24 EP disclosed
WO-2002051923-A2 METHOD FOR REDUCING HAZE IN A FIRE RESISTANT POLYCARBONATE COMPOSITION GENERAL ELECTRIC COMPANY (US) 2002-07-04 WO disclosed
US-4174359-A HALOGEN COMPOUND MOBAY CHEMICAL CORPORATION (US) 1979-11-13 US disclosed