SCHEMBL7280147

SCHEMBL7280147

O=C(OCc1ccncc1)c1c[nH]c2ccccc12

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 1/20 0.55
NR4A2 P43354 2/20 0.55
CREBBP Q92793 1/20 0.55
LMNA P02545 1/20 0.52
ALDH1A1 P00352 2/20 0.51
RAB9A P51151 2/20 0.51
CYP1A2 P05177 1/20 0.51
CYP2D6 P10635 1/20 0.51
CYP2C9 P11712 1/20 0.51
TSHR P16473 1/20 0.51
THPO P40225 1/20 0.51
PMP22 Q01453 1/20 0.50
GPR84 Q9NQS5 1/20 0.50
ATM Q13315 2/20 0.48
PBRM1 Q86U86 1/20 0.48
L3MBTL1 Q9Y468 1/20 0.47
NPC1 O15118 1/20 0.47
MEN1 O00255 1/20 0.47
MAPT P10636 1/20 0.47
KMT2A Q03164 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3264030 0.89 NR4A2 (0.61) NR4A2CREBBPLMNAALDH1A1RAB9A
SCHEMBL7280152 0.86 NR4A2 (0.51) NR4A2CREBBPLMNAALDH1A1RAB9A
SCHEMBL7280001 0.80 HTR2C (0.58) NR4A2CREBBPLMNAALDH1A1RAB9A
SCHEMBL730525 0.77 NR4A2 (0.69) NR4A2CREBBPLMNAALDH1A1RAB9A
SCHEMBL14793753 0.76 TDP1 (0.52) NR4A2LMNAALDH1A1RAB9AKMT2A
SCHEMBL7835246 0.76 TDP1 (0.52) NR4A2LMNAALDH1A1CYP2C9TSHR
Hydrochloric Acid SCHEMBL30718988 0.76 NR4A2 (0.67) NR4A2CREBBPLMNAALDH1A1RAB9A
Hydrochloric Acid SCHEMBL28308377 0.76 NR4A2 (0.67) NR4A2CREBBPLMNAALDH1A1RAB9A
SCHEMBL7636009 0.75 GABRA1 (0.60) NR4A2CREBBPLMNARAB9AGPR84
SCHEMBL5805847 0.74 NR4A2 (0.65) NR4A2CREBBPLMNAALDH1A1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0429984-B1 Indole derivatives NISSHIN FLOUR MILLING CO (JP) 1997-07-23 EP disclosed
US-5124324-A Psychological disorders, 5-hydroxy tryptamine antagonists NISSHIN FLOUR MILLING CO., LTD. (JP) 1992-06-23 US disclosed
EP-0429984-A2 Indole derivatives NISSHIN FLOUR MILLING CO., LTD. (JP) 1991-06-05 EP disclosed